Endomorphin-2: a biased agonist at the μ-opioid receptor. (Q36105495)

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31 January 2020

title

Endomorphin-2: a biased agonist at the μ-opioid receptor (English)

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31 January 2020

1

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Craig A McArdle

6

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31 January 2020

Elizabeth M Rosethorne

7

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31 January 2020

Steven J. Charlton

8

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31 January 2020

Cornelius Krasel

9

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31 January 2020

Chris Bailey

10

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31 January 2020

author name string

Javier Llorente

2

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31 January 2020

Jamie McPherson

3

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31 January 2020

Alex Cooke

4

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31 January 2020

Stuart J Mundell

5

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31 January 2020

Graeme Henderson

11

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31 January 2020

Eamonn Kelly

12

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publication date

2 May 2012

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31 January 2020

published in

Molecular Pharmacology

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31 January 2020

volume

82

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31 January 2020

issue

2

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31 January 2020

page(s)

178-188

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Molecular mechanism of β-arrestin-biased agonism at seven-transmembrane receptors

31 January 2020

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2 October 2017

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Search of the human proteome for endomorphin-1 and endomorphin-2 precursor proteins.

2 October 2017

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2 October 2017

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2 October 2017

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Activation and internalization of the mu-opioid receptor by the newly discovered endogenous agonists, endomorphin-1 and endomorphin-2

2 October 2017

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Endomorphin-1 and endomorphin-2 are partial agonists at the human mu-opioid receptor

2 October 2017

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Specific G protein activation and mu-opioid receptor internalization caused by morphine, DAMGO and endomorphin I

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23 September 2018

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23 September 2018

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23 September 2018

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Receptor constants for endomorphin-1 and endomorphin-1-ol indicate differences in efficacy and receptor occupancy

23 September 2018

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23 September 2018

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Characterization of endomorphin-1 and -2 on [35S]GTPgammaS binding in the mouse spinal cord.

23 September 2018

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Endomorphin-stimulated [35S]GTPgammaS binding in rat brain: evidence for partial agonist activity at mu-opioid receptors.

23 September 2018

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On the potassium conductance increased by opioids in rat locus coeruleus neurones

23 September 2018

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23 September 2018

Identifiers

DOI

10.1124/MOL.112.078659

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31 January 2020

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31 January 2020

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