Novel Noncatalytic Substrate-Selective p38α-Specific MAPK Inhibitors with Endothelial-Stabilizing and Anti-Inflammatory Activity. (Q42380665)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:28298524%20AND%20SRC:MED&resulttype=core&format=json

6 April 2020

title

Novel Noncatalytic Substrate-Selective p38α-Specific MAPK Inhibitors with Endothelial-Stabilizing and Anti-Inflammatory Activity (English)

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6 April 2020

6

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6 April 2020

Ramin Samadani

8

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6 April 2020

Alex MacKerell

10

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6 April 2020

author name string

Nirav G Shah

1

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6 April 2020

Mohan E Tulapurkar

2

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6 April 2020

Aparna Ramarathnam

3

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6 April 2020

Amanda Brophy

4

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6 April 2020

Ramon Martinez

5

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6 April 2020

Theresa Hodges

7

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6 April 2020

Ishwar S Singh

9

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6 April 2020

Paul Shapiro

11

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6 April 2020

Jeffrey D Hasday

12

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6 April 2020

language of work or name

English

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publication date

15 March 2017

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6 April 2020

published in

Journal of Immunology

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6 April 2020

volume

198

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6 April 2020

issue

8

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6 April 2020

page(s)

3296-3306

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describes a project that uses

6 April 2020

ImageQuant

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11 June 2022

https://www.ebi.ac.uk/europepmc/webservices/rest/PMC5649369/fullTextXML

inferred from PubMed Central ID database lookup

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28 May 2018

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28 May 2018

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28 May 2018

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28 May 2018

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Inhibition of p38 mitogen-activated protein kinase improves nitric oxide-mediated vasodilatation and reduces inflammation in hypercholesterolemia.

16 August 2018

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16 August 2018

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16 August 2018

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16 August 2018

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Mobilization of neutrophil sialidase activity desialylates the pulmonary vascular endothelial surface and increases resting neutrophil adhesion to and migration across the endothelium

16 August 2018

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Consideration of molecular weight during compound selection in virtual target-based database screening

16 August 2018

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16 August 2018

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16 August 2018

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Crossref

https://api.crossref.org/works/10.4049%2FJIMMUNOL.1602059

Binding Response: A Descriptor for Selecting Ligand Binding Site on Protein Surfaces

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.4049%2FJIMMUNOL.1602059

Oral p38 mitogen-activated protein kinase inhibition with BIRB 796 for active Crohn's disease: a randomized, double-blind, placebo-controlled trial

21 January 2018

1 reference

12 December 2020

TNF induces distinct gene expression programs in microvascular and macrovascular human endothelial cells

1 reference

12 December 2020

Pharmacological profile of SB 203580, a selective inhibitor of cytokine suppressive binding protein/p38 kinase, in animal models of arthritis, bone resorption, endotoxin shock and immune function

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12 December 2020

Chemical genetics define the roles of p38alpha and p38beta in acute and chronic inflammation

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12 December 2020

Anatomy of fingerprint search calculations on structurally diverse sets of active compounds

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12 December 2020

Identifiers

DOI

10.4049/JIMMUNOL.1602059

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:28298524%20AND%20SRC:MED&resulttype=core&format=json

6 April 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:28298524%20AND%20SRC:MED&resulttype=core&format=json

6 April 2020

1 reference