Ligand-enabled β-C-H arylation of α-amino acids using a simple and practical auxiliary (Q40701143)

22 September 2017

Ligand-enabled β-C-H arylation of α-amino acids using a simple and practical auxiliary (English)

1 reference

22 September 2017

Jian He

6

0 references

Jin-Quan Yu

13

object named as

Jin-Quan Yu

1 reference

22 September 2017

Gang Chen

1

1 reference

22 September 2017

Toshihiko Shigenari

2

1 reference

22 September 2017

Pankaj Jain

3

1 reference

22 September 2017

Zhipeng Zhang

4

1 reference

22 September 2017

Zhong Jin

5

1 reference

22 September 2017

Suhua Li

7

1 reference

22 September 2017

Claudio Mapelli

8

1 reference

22 September 2017

Michael M Miller

9

1 reference

22 September 2017

Michael A Poss

10

1 reference

22 September 2017

Paul M Scola

11

1 reference

22 September 2017

Kap-Sun Yeung

12

1 reference

22 September 2017

language of work or name

English

0 references

publication date

3 March 2015

1 reference

Journal of the American Chemical Society

22 September 2017

1 reference

22 September 2017

137

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22 September 2017

9

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22 September 2017

3338-3351

1 reference

Structure-Based Design of Irreversible Human KAT II Inhibitors: Discovery of New Potency-Enhancing Interactions

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Discovery of Brain-Penetrant, Irreversible Kynurenine Aminotransferase II Inhibitors for Schizophrenia.

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Palladium(II)-catalyzed enantioselective C(sp³)-H activation using a chiral hydroxamic acid ligand

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Ligand-enabled methylene C(sp3)-H bond activation with a Pd(II) catalyst

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Biotinylated Rh(III) complexes in engineered streptavidin for accelerated asymmetric C-H activation

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Fragment screening at adenosine-A(3) receptors in living cells using a fluorescence-based binding assay

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Analogues of doxanthrine reveal differences between the dopamine D1 receptor binding properties of chromanoisoquinolines and hexahydrobenzo[a]phenanthridines

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Pd(II)-catalyzed enantioselective C-H activation of cyclopropanes

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Pd(II)-catalyzed olefination of sp3 C-H bonds

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Auxiliary-assisted palladium-catalyzed arylation and alkylation of sp2 and sp3 carbon-hydrogen bonds

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Pd(0)/PR3-catalyzed intermolecular arylation of sp3 C-H bonds

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Palladium- and copper-catalyzed arylation of carbon-hydrogen bonds

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Comparison of the enantiomers of (+/-)-doxanthrine, a high efficacy full dopamine D(1) receptor agonist, and a reversal of enantioselectivity at D(1) versus alpha(2C) adrenergic receptors

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Rational design, synthesis, biologic evaluation, and structure-activity relationship studies of novel 1-indanone alpha(1)-adrenoceptor antagonists

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

trans-2,3-dihydroxy-6a,7,8,12b-tetrahydro-6H-chromeno[3,4-c]isoquinoline: synthesis, resolution, and preliminary pharmacological characterization of a new dopamine D1 receptor full agonist

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Development of potent, orally active 1-substituted-3,4-dihydro-2-quinolone glycogen phosphorylase inhibitors

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Phosphoramidites: marvellous ligands in catalytic asymmetric conjugate addition

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Synthesis and antibacterial activities of some chloro analogs of 3-amino-3,4-dihydro-1-hydroxycarbostyril

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Generation of N-methyl-D-aspartate agonist and competitive antagonist pharmacophore models. Design and synthesis of phosphonoalkyl-substituted tetrahydroisoquinolines as novel antagonists

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Overcoming the limitations of directed C-H functionalizations of heterocycles

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Nonnatural amino acid synthesis by using carbon-hydrogen bond functionalization methodology

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Total synthesis of celogentin C by stereoselective C-H activation.

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

The mechanism of a ligand-promoted C(sp3)-H activation and arylation reaction via palladium catalysis: theoretical demonstration of a Pd(II)/Pd(IV) redox manifold.

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Ligand-promoted alkylation of C(sp3)-H and C(sp2)-H bonds

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Ligand-controlled C(sp³)-H arylation and olefination in synthesis of unnatural chiral α-amino acids

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Nickel-catalyzed chelation-assisted direct arylation of unactivated C(sp3)-H bonds with aryl halides.

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Nickel-catalyzed direct arylation of C(sp3)-H bonds in aliphatic amides via bidentate-chelation assistance.

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Direct conversion of N-alkoxyamides to carboxylic esters through tandem NBS-mediated oxidative homocoupling and thermal denitrogenation

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Chiral cyclopentadienyl ligands as stereocontrolling element in asymmetric C-H functionalization.

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Organocatalytic, oxidative, intermolecular amination and hydrazination of simple arenes at ambient temperature.

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Understanding reactivity and stereoselectivity in palladium-catalyzed diastereoselective sp3 C-H bond activation: intermediate characterization and computational studies.

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Ruthenium-catalyzed C-H/N-O bond functionalization: green isoquinolone syntheses in water.

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Facile benzo-ring construction via palladium-catalyzed functionalization of unactivated sp3 C-H bonds under mild reaction conditions

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Rhodium(III)-catalyzed isoquinolone synthesis: the N-O bond as a handle for C-N bond formation and catalyst turnover

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Synthesis of beta-, gamma-, and delta-lactams via Pd(II)-catalyzed C-H activation reactions

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Pd(II)-catalyzed cross-coupling of sp3 C-H Bonds with sp2 and sp3 boronic acids using air as the oxidant

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Highly regioselective arylation of sp3 C-H bonds catalyzed by palladium acetate

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Palladium-catalyzed oxygenation of unactivated sp3 C-H bonds

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

New chiral phosphorus ligands for enantioselective hydrogenation.

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

One-Pot Formation of CC and CN Bonds through Palladium-Catalyzed Dual CH Activation: Synthesis of Phenanthridinones

19 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

Rh(III)-Catalyzed Directed C−H Olefination Using an Oxidizing Directing Group: Mild, Efficient, and Versatile

2 December 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4432912

SYNTHESIS AND MICROBIOLOGICAL PROPERTIES OF 3-AMINO-3,4-DIHYDRO-1-HYDROXYCARBOSTYRIL

2 December 2018

1 reference

12 December 2020

β-Arylation of carboxamides via iron-catalyzed C(sp3)-H bond activation

1 reference

12 December 2020

Catalytic, asymmetric, and stereodivergent synthesis of non-symmetric β,β-diaryl-α-amino acids

1 reference

12 December 2020

Synthesis of Indolines via Pd(II)-Catalyzed Amination of C–H Bonds Using PhI(OAc)2as the Bystanding Oxidant

1 reference

12 December 2020

Copper-catalyzed site-selective intramolecular amidation of unactivated C(sp³)-H bonds

1 reference

12 December 2020

Pyridine-2,6-bis(oxazolines), helpful ligands for asymmetric catalysts

1 reference

12 December 2020

Cu-catalyzed asymmetric conjugate additions of alkylzinc reagents to acyclic aliphatic enones

1 reference

12 December 2020

Novel acetoxylation and C-C coupling reactions at unactivated positions in alpha-amino acid derivatives

1 reference

12 December 2020

Palladium-catalyzed asymmetric iodination of unactivated C-H bonds under mild conditions

1 reference

12 December 2020

Synthesis of phenanthridinones from N-methoxybenzamides and arenes by multiple palladium-catalyzed C-H activation steps at room temperature

1 reference

12 December 2020

Solid phase synthesis of peptides containing the non-hydrolysable analog of (O)phosphotyrosine, p(CH2PO3H2)Phe. Application to the synthesis of 344-357 sequences of the beta 2 adrenergic receptor

1 reference

12 December 2020

Ruthenium-catalyzed isoquinolone synthesis through C-H activation using an oxidizing directing group

1 reference

12 December 2020

Copper-catalyzed intramolecular C(sp³)-H and C(sp²)-H amidation by oxidative cyclization

1 reference

12 December 2020

Rhodium-catalyzed asymmetric 1,4-addition and its related asymmetric reactions

1 reference

12 December 2020

Stereoselective Synthesis of Chiral α-Amino-β-Lactams through Palladium(II)-Catalyzed Sequential Monoarylation/Amidation of C(sp3)H Bonds

1 reference

12 December 2020

Highly selective mild stepwise allylation of N-methoxybenzamides with allenes

1 reference

12 December 2020

A general strategy for the synthesis of cyclic N-aryl hydroxamic acids via partial nitro group reduction

1 reference

12 December 2020

Ruthenium-catalyzed oxidative C-H bond olefination of N-methoxybenzamides using an oxidizing directing group

1 reference

12 December 2020

Pd-catalysed synthesis of isoquinolinones and analogues via C-H and N-H bonds double activation

1 reference

12 December 2020

Tetrapeptide tyrosine kinase inhibitors. Enantioselective synthesis of p-hydroxymethyl-L-phenylalanine, incorporation into a tetrapeptide, and subsequent elaboration into p-(R,S-hydroxyphosphonomethyl)-L-phenylalanine

1 reference

12 December 2020

Pd-catalyzed stereoselective oxidation of methyl groups by inexpensive oxidants under mild conditions: a dual role for carboxylic anhydrides in catalytic C--H bond oxidation

1 reference

12 December 2020

Nickel-catalyzed site-selective alkylation of unactivated C(sp3)-H bonds

1 reference

12 December 2020

Palladium-Catalyzed Methylation and Arylation of sp2and sp3C−H Bonds in Simple Carboxylic Acids

1 reference

12 December 2020

New Heteroannulation Reactions ofN-Alkoxybenzamides by Pd(II) Catalyzed C–H Activation

1 reference

12 December 2020

A general and practical palladium-catalyzed monoarylation of β-methyl C(sp3)–H of alanine

1 reference

12 December 2020

Identifiers

DOI

10.1021/JA512690X

1 reference

22 September 2017

1 reference

22 September 2017

1 reference