New class of HIV integrase inhibitors that block viral replication in cell culture (Q40639670)

22 September 2017

New class of HIV integrase inhibitors that block viral replication in cell culture (English)

1 reference

22 September 2017

8

Zeger Debyser

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Bénédicte Van Maele

3

Bénédicte Van Maele

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Victor V. Tetz

Victor Tetz

4

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Christophe Pannecouque

Christophe Pannecouque

1

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Erik De Clercq

Erik De Clercq

6

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Myriam Witvrouw

7

Myriam Witvrouw

1 reference

22 September 2017

2

Wim Pluymers

1 reference

22 September 2017

5

Peter Cherepanov

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PubMed ID

12176326

22 September 2017

language of work or name

English

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publication date

1 July 2002

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22 September 2017

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22 September 2017

12

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22 September 2017

14

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22 September 2017

1169-1177

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New developments in anti-HIV chemotherapy

22 September 2017

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

1 reference

7 January 2021

Requirement of active human immunodeficiency virus type 1 integrase enzyme for productive infection of human T-lymphoid cells

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

HIV-1 integration as a target for antiretroviral therapy: a review

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Reversal of Integration and DNA Splicing Mediated by Integrase of Human Immunodeficiency Virus

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Repair of gaps in retroviral DNA integration intermediates

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Modeling the late steps in HIV-1 retroviral integrase-catalyzed DNA integration

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

A high-throughput, non-radioactive microtiter plate assay for activity of the human immunodeficiency virus integrase protein

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

A novel assay for the DNA strand-transfer reaction of HIV-1 integrase

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Differential inhibition of HIV-1 preintegration complexes and purified integrase protein by small molecules

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Human immunodeficiency virus integration protein expressed in Escherichia coli possesses selective DNA cleaving activity

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Activities of human immunodeficiency virus (HIV) integration protein in vitro: specific cleavage and integration of HIV DNA

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Retroviral integrase inhibitors year 2000: update and perspectives

1 reference

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7 January 2021

HIV-1 integrase inhibitors: past, present, and future

1 reference

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7 January 2021

T30177, an oligonucleotide stabilized by an intramolecular guanosine octet, is a potent inhibitor of laboratory strains and clinical isolates of human immunodeficiency virus type 1

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Mode of interaction of G-quartets with the integrase of human immunodeficiency virus type 1.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Human immunodeficiency virus glycoprotein gp120 as the primary target for the antiviral action of AR177 (Zintevir).

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Inhibitors of HIV-1 replication [corrected; erratum to be published] that inhibit HIV integrase

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Resistance to the anti-human immunodeficiency virus type 1 compound L-chicoric acid results from a single mutation at amino acid 140 of integrase

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Inhibition of HIV-1 integrase by flavones, caffeic acid phenethyl ester (CAPE) and related compounds

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Effects of Tyrphostins, Protein Kinase Inhibitors, on Human Immunodeficiency Virus Type 1 Integrase

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

(-)-Arctigenin as a lead structure for inhibitors of human immunodeficiency virus type-1 integrase

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Hydroxylated aromatic inhibitors of HIV-1 integrase

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Inhibition of human immunodeficiency virus type-1 integrase by curcumin

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Antiretroviral agents as inhibitors of both human immunodeficiency virus type 1 integrase and protease.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Potent inhibitors of human immunodeficiency virus type 1 integrase: identification of a novel four-point pharmacophore and tetracyclines as novel inhibitors.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Inhibitors of human immunodeficiency virus integrase

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Inhibition of the in vitro integration of Moloney murine leukemia virus DNA by the DNA minor groove binder netropsin

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Alternate strand DNA triple helix-mediated inhibition of HIV-1 U5 long terminal repeat integration in vitro

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Peptide inhibitors of HIV-1 integrase dissociate the enzyme oligomers

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Structure-activity relationships and binding mode of styrylquinolines as potent inhibitors of HIV-1 integrase and replication of HIV-1 in cell culture

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Thiazolothiazepine inhibitors of HIV-1 integrase

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Inhibitors of strand transfer that prevent integration and inhibit HIV-1 replication in cells

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

Structure of the HIV-1 integrase catalytic domain complexed with an inhibitor: a platform for antiviral drug design

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

4-Aryl-2,4-dioxobutanoic acid inhibitors of HIV-1 integrase and viral replication in cells

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

In vivo gene delivery and stable transduction of nondividing cells by a lentiviral vector

1 reference

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7 January 2021

Multiply attenuated lentiviral vector achieves efficient gene delivery in vivo

1 reference

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7 January 2021

An antiviral target on reverse transcriptase of human immunodeficiency virus type 1 revealed by tetrahydroimidazo-[4,5,1-jk] [1,4]benzodiazepin-2 (1H)-one and -thione derivatives

1 reference

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7 January 2021

A two plasmid co-expression system in Escherichia coli for the production of virion-like reverse transcriptase of the human immunodeficiency virus type 1.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

A quantitative assay for HIV DNA integration in vivo

1 reference

https://api.crossref.org/works/10.1016%2FS0960-9822%2802%2900952-1

7 January 2021

10.1016/S0960-9822(02)00952-1

Identifiers

DOI

1 reference

22 September 2017

1 reference

PubMed ID

12176326