Influence of ligand binding kinetics on functional inhibition of human recombinant serotonin and norepinephrine transporters (Q39758568)

14 September 2017

Influence of ligand binding kinetics on functional inhibition of human recombinant serotonin and norepinephrine transporters (English)

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14 September 2017

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William J Martin

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author name string

Pamela R Tsuruda

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14 September 2017

Joey Yung

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14 September 2017

Ray Chang

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14 September 2017

Ngoc Mai

5

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14 September 2017

Jacqueline A M Smith

6

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14 September 2017

28 December 2009

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Journal of Pharmacological and Toxicological Methods

14 September 2017

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14 September 2017

61

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14 September 2017

2

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14 September 2017

192-204

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A new look at the statistical model identification

14 September 2017

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https://api.crossref.org/works/10.1016%2FJ.VASCN.2009.12.003

Location of the antidepressant binding site in the serotonin transporter: importance of Ser-438 in recognition of citalopram and tricyclic antidepressants.

7 January 2021

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Antidepressants targeting the serotonin reuptake transporter act via a competitive mechanism

7 January 2021

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The binding sites for cocaine and dopamine in the dopamine transporter overlap

7 January 2021

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

7 January 2021

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https://api.crossref.org/works/10.1016%2FJ.VASCN.2009.12.003

Binding characteristics of selective serotonin reuptake inhibitors with relation to emission tomography studies

7 January 2021

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Comparative evaluation in nonhuman primates of five PET radiotracers for imaging the serotonin transporters: [11C]McN 5652, [11C]ADAM, [11C]DASB, [11C]DAPA, and [11C]AFM.

7 January 2021

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https://api.crossref.org/works/10.1016%2FJ.VASCN.2009.12.003

Validation of a fluorescence-based high-throughput assay for the measurement of neurotransmitter transporter uptake activity

7 January 2021

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Differential inhibitory effects of drugs acting at the noradrenaline and 5-hydroxytryptamine transporters in rat and human neocortical synaptosomes

7 January 2021

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https://api.crossref.org/works/10.1016%2FJ.VASCN.2009.12.003

Kinetic and thermodynamic assessment of binding of serotonin transporter inhibitors

7 January 2021

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https://api.crossref.org/works/10.1016%2FJ.VASCN.2009.12.003

Desvenlafaxine succinate identifies novel antagonist binding determinants in the human norepinephrine transporter

7 January 2021

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Identification and characterization of pseudoirreversible nonpeptide antagonists of the neuropeptide Y Y5 receptor and development of a novel Y5-selective radioligand

7 January 2021

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Studies of the biogenic amine transporters. XI. Identification of a 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine (GBR12909) analog that allosterically modulates the serotonin transporter

7 January 2021

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The kinetics of action of acetylcholine antagonists in smooth muscle

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The molecular mechanism of "ecstasy" [3,4-methylenedioxy-methamphetamine (MDMA)]: serotonin transporters are targets for MDMA-induced serotonin release

7 January 2021

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Antidepressant binding site in a bacterial homologue of neurotransmitter transporters

7 January 2021

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SNRIs: The Pharmacology, Clinical Efficacy, and Tolerability in Comparison with Other Classes of Antidepressants

7 January 2021

1 reference

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Fluoxetine (Prozac) binding to serotonin transporter is modulated by chloride and conformational changes

7 January 2021

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Plasma membrane monoamine transporters: structure, regulation and function

7 January 2021

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Milnacipran: a comparative analysis of human monoamine uptake and transporter binding affinity

7 January 2021

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Sartan-AT1 receptor interactions: in vitro evidence for insurmountable antagonism and inverse agonism

7 January 2021

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LeuT-desipramine structure reveals how antidepressants block neurotransmitter reuptake

7 January 2021

1 reference

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Antidepressant specificity of serotonin transporter suggested by three LeuT-SSRI structures

7 January 2021

1 reference

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10.1016/J.VASCN.2009.12.003

7 January 2021

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14 September 2017

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