A selective TSH receptor antagonist inhibits stimulation of thyroid function in female mice (Q37405158)

20 August 2017

A selective TSH receptor antagonist inhibits stimulation of thyroid function in female mice (English)

1 reference

20 August 2017

Susanne Neumann

1

1 reference

20 August 2017

Eshel A Nir

2

1 reference

20 August 2017

Elena Eliseeva

3

1 reference

20 August 2017

Wenwei Huang

4

1 reference

20 August 2017

Juan Marugan

5

1 reference

20 August 2017

Jingbo Xiao

6

1 reference

20 August 2017

Andrés E Dulcey

7

1 reference

20 August 2017

Marvin C Gershengorn

8

1 reference

20 August 2017

language of work or name

English

0 references

publication date

4 December 2013

1 reference

20 August 2017

1 reference

20 August 2017

155

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20 August 2017

1

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20 August 2017

310-314

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A small molecule antagonist inhibits thyrotropin receptor antibody-induced orbital fibroblast functions involved in the pathogenesis of Graves ophthalmopathy

20 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

Update in TSH receptor agonists and antagonists

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

A drug-like antagonist inhibits thyrotropin receptor-mediated stimulation of cAMP production in Graves' orbital fibroblasts

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

Mechanism of action of a nanomolar potent, allosteric antagonist of the thyroid-stimulating hormone receptor

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

A new small-molecule antagonist inhibits Graves' disease antibody activation of the TSH receptor

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

Variable suppression of serum thyroxine in female mice of different inbred strains by triiodothyronine administered in drinking water

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

A small molecule inverse agonist for the human thyroid-stimulating hormone receptor

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

6 September 2017

Graves' ophthalmopathy

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

Small-molecule agonists for the thyrotropin receptor stimulate thyroid function in human thyrocytes and mice

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

Thyrotropin and homologous glycoprotein hormone receptors: structural and functional aspects of extracellular signaling mechanisms

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

A low-molecular-weight antagonist for the human thyrotropin receptor with therapeutic potential for hyperthyroidism

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

Thyrotropin receptor-associated diseases: from adenomata to Graves disease

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

Complete inhibition of rhTSH-, Graves' disease IgG-, and M22-induced cAMP production in differentiated orbital fibroblasts by a low-molecular-weight TSHR antagonist

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

TSH receptor monoclonal antibodies with agonist, antagonist, and inverse agonist activities.

2 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

Suppression of thyrotropin receptor constitutive activity by a monoclonal antibody with inverse agonist activity.

2 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

Human monoclonal thyroid stimulating autoantibody.

2 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868809

Development of ALZET® osmotic pump compatible solvent compositions to solubilize poorly soluble compounds for preclinical studies

2 September 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24169564

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

When will thyrotropin receptor antagonists and inverse thyrotropin receptor agonists become available for clinical use?

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24169564

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1210/EN.2013-1835

1 reference

20 August 2017

1 reference

20 August 2017

1 reference