The binding sites for benztropines and dopamine in the dopamine transporter overlap. (Q36990361)

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13 February 2020

title

The binding sites for benztropines and dopamine in the dopamine transporter overlap (English)

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13 February 2020

0 references

6

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Lei Shi

7

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Claus J Loland

8

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Ulrik Gether

9

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author name string

Heidi Bisgaard

1

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13 February 2020

M Andreas B Larsen

2

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Sonia Mazier

3

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Thijs Beuming

4

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Amy Hauck Newman

5

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publication date

6 September 2010

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13 February 2020

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13 February 2020

volume

60

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page(s)

182-190

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issue

1

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Substrate-dependent proton antiport in neurotransmitter:sodium symporters

13 February 2020

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4 September 2018

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4 September 2018

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Identification of intracellular residues in the dopamine transporter critical for regulation of transporter conformation and cocaine binding.

4 September 2018

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Evaluation of the blood-brain barrier transport, population pharmacokinetics, and brain distribution of benztropine analogs and cocaine using in vitro and in vivo techniques

4 September 2018

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4 September 2018

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Defining proximity relationships in the tertiary structure of the dopamine transporter. Identification of a conserved glutamic acid as a third coordinate in the endogenous Zn(2+)-binding site.

4 September 2018

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4 September 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/20816875

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Population Pharmacokinetics, Brain Distribution, and Pharmacodynamics of 2nd Generation Dopamine Transporter Selective Benztropine Analogs Developed as Potential Substitute Therapeutics for Treatment of Cocaine Abuse

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20816875

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

An intracellular interaction network regulates conformational transitions in the dopamine transporter.

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20816875

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.NEUROPHARM.2010.08.021

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20816875%20AND%20SRC:MED&resulttype=core&format=json

13 February 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20816875%20AND%20SRC:MED&resulttype=core&format=json

13 February 2020

1 reference