GABAB receptor-positive modulators: brain region-dependent effects (Q35650701)

9 August 2017

GABAB receptor-positive modulators: brain region-dependent effects (English)

1 reference

9 August 2017

Julie G Hensler

1

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9 August 2017

Tushar Advani

2

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9 August 2017

Teresa F Burke

3

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9 August 2017

Kejun Cheng

4

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9 August 2017

Kenner C Rice

5

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9 August 2017

Wouter Koek

6

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9 August 2017

language of work or name

English

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publication date

27 September 2011

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Journal of Pharmacology and Experimental Therapeutics

9 August 2017

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9 August 2017

340

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9 August 2017

1

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9 August 2017

19-26

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describes a project that uses

9 August 2017

ImageJ

1 reference

11 June 2022

https://www.ebi.ac.uk/europepmc/webservices/rest/PMC3251019/fullTextXML

based on heuristic

inferred from PubMed Central ID database lookup

cites work

GABAB receptors in reward processes

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GABAB receptors: physiological functions and mechanisms of diversity

12 July 2018

1 reference

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GABAB receptor-positive modulators: enhancement of GABAB receptor agonist effects in vivo

12 July 2018

1 reference

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Native GABA(B) receptors are heteromultimers with a family of auxiliary subunits

12 July 2018

1 reference

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Role of the GABA(B) receptor system in alcoholism and stress: focus on clinical studies and treatment perspectives

12 July 2018

1 reference

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Allosteric modulators of GABA(B) receptors: mechanism of action and therapeutic perspective.

12 July 2018

1 reference

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Allosteric modulators of GPCRs: a novel approach for the treatment of CNS disorders

12 July 2018

1 reference

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Behavioral analyses of GHB: receptor mechanisms

12 July 2018

1 reference

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Characterization of (R,S)-5,7-di-tert-butyl-3-hydroxy-3-trifluoromethyl-3H-benzofuran-2-one as a positive allosteric modulator of GABAB receptors

12 July 2018

1 reference

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CGP7930: a positive allosteric modulator of the GABAB receptor.

12 July 2018

1 reference

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Dominant role of GABAB2 and Gbetagamma for GABAB receptor-mediated-ERK1/2/CREB pathway in cerebellar neurons.

12 July 2018

1 reference

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GABAB receptor: a site of therapeutic benefit

12 July 2018

1 reference

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Mechanisms of allosteric modulation at GABAB receptors by CGP7930 and GS39783: effects on affinities and efficacies of orthosteric ligands with distinct intrinsic properties.

12 July 2018

1 reference

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Don't worry 'B' happy!: a role for GABA(B) receptors in anxiety and depression.

12 July 2018

1 reference

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Gamma-hydroxybutyric acid (GHB) and gamma-aminobutyric acidB receptor (GABABR) binding sites are distinctive from one another: molecular evidence.

12 July 2018

1 reference

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In vivo effectiveness of CGP7930, a positive allosteric modulator of the GABAB receptor

12 July 2018

1 reference

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Molecular structure and physiological functions of GABA(B) receptors

12 July 2018

1 reference

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Allosteric modulation of G-protein coupled receptors.

12 July 2018

1 reference

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Effects of GABA agonists on body temperature regulation in GABA(B(1))-/- mice

12 July 2018

1 reference

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GABA(B) receptors: from monogamy to promiscuity

12 July 2018

1 reference

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International Union of Pharmacology. XXXIII. Mammalian gamma-aminobutyric acid(B) receptors: structure and function

12 July 2018

1 reference

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Positive allosteric modulation of native and recombinant gamma-aminobutyric acid(B) receptors by 2,6-Di-tert-butyl-4-(3-hydroxy-2,2-dimethyl-propyl)-phenol (CGP7930) and its aldehyde analog CGP13501

12 July 2018

1 reference

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Regulation of 5-HT(1A) receptor-stimulated [35S]-GtpgammaS binding as measured by quantitative autoradiography following chronic agonist administration

12 July 2018

1 reference

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GABA(B) receptor activation of Purkinje cells in cerebellar slices.

12 July 2018

1 reference

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Relation of the [3H] gamma-hydroxybutyric acid (GHB) binding site to the gamma-aminobutyric acidB (GABAB) receptor in rat brain

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3251019

A physiological role for GABAB receptors and the effects of baclofen in the mammalian central nervous system

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3251019

GABAB receptor activation protects neurons from apoptosis via IGF-1 receptor transactivation.

12 July 2018

1 reference

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Specific reduction of alcohol's motivational properties by the positive allosteric modulator of the GABAB receptor, GS39783--comparison with the effect of the GABAB receptor direct agonist, baclofen

25 September 2018

1 reference

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Cataleptic effects of gamma-hydroxybutyrate (GHB), its precursor gamma-butyrolactone (GBL), and GABAB receptor agonists in mice: differential antagonism by the GABAB receptor antagonist CGP35348.

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3251019

Effect of early rearing conditions on alcohol drinking and 5-HT1A receptor function in C57BL/6J mice.

25 September 2018

1 reference

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Novel gamma-hydroxybutyric acid (GHB) analogs share some, but not all, of the behavioral effects of GHB and GABAB receptor agonists

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3251019

Specific gamma-hydroxybutyrate-binding sites but loss of pharmacological effects of gamma-hydroxybutyrate in GABA(B)(1)-deficient mice

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3251019

Quantitative autoradiographic analysis of the new radioligand [(3)H](2E)-(5-hydroxy-5,7,8,9-tetrahydro-6H-benzo[a][7]annulen-6-ylidene) ethanoic acid ([(3)H]NCS-382) at gamma-hydroxybutyric acid (GHB) binding sites in rat brain

25 September 2018

1 reference

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Gamma-hydroxybutyrate is a weak agonist at recombinant GABA(B) receptors.

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3251019

Binding characteristics of gamma-hydroxybutyric acid as a weak but selective GABAB receptor agonist.

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3251019

Distribution and kinetics of GABAB binding sites in rat central nervous system: a quantitative autoradiographic study

25 September 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21954301

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Distribution of the auxiliary GABAB receptor subunits KCTD8, 12, 12b, and 16 in the mouse brain

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21954301

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1124/JPET.111.186577

1 reference

9 August 2017

1 reference

9 August 2017

1 reference