Analysis of transmembrane domains 1 and 4 of the human angiotensin II AT1 receptor by cysteine-scanning mutagenesis (Q33593826)

28 July 2017

title

Analysis of transmembrane domains 1 and 4 of the human angiotensin II AT1 receptor by cysteine-scanning mutagenesis (English)

1 reference

28 July 2017

main subject

transmembrane protein

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Emanuel Escher

4

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author name string

Liping Yan

1

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28 July 2017

Brian J Holleran

2

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28 July 2017

Pierre Lavigne

3

1 reference

28 July 2017

Gaétan Guillemette

5

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28 July 2017

Richard Leduc

6

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28 July 2017

language of work or name

English

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publication date

23 November 2009

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Journal of Biological Chemistry

28 July 2017

published in

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28 July 2017

volume

285

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28 July 2017

issue

4

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28 July 2017

page(s)

2284-2293

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The second transmembrane domain of the human type 1 angiotensin II receptor participates in the formation of the ligand binding pocket and undergoes integral pivoting movement during the process of receptor activation

28 July 2017

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Analysis of the third transmembrane domain of the human type 1 angiotensin II receptor by cysteine scanning mutagenesis

21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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Mechanism of constitutive activation of the AT1 receptor: influence of the size of the agonist switch binding residue Asn(111).

21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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The fifth transmembrane domain of angiotensin II Type 1 receptor participates in the formation of the ligand-binding pocket and undergoes a counterclockwise rotation upon receptor activation

21 January 2018

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Mutagenesis of the AT1 receptor reveals different binding modes of angiotensin II and [Sar1]-angiotensin II.

21 January 2018

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21 January 2018

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30 October 2018

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30 October 2018

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Role of transmembrane helix IV in G-protein specificity of the angiotensin II type 1 receptor

21 January 2018

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12 December 2020

Identification of residues involved in ligand binding to the neurokinin-2 receptor

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12 December 2020

A computer modeling postulated mechanism for angiotensin II receptor activation

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12 December 2020

Substituted-cysteine accessibility method

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12 December 2020

Conformational changes in rhodopsin. Movement of helix f detected by site-specific chemical labeling and fluorescence spectroscopy

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12 December 2020

Activation of the angiotensin II type 1 receptor leads to movement of the sixth transmembrane domain: analysis by the substituted cysteine accessibility method

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12 December 2020

Novel aromatic residues in transmembrane domains IV and V involved in agonist binding at alpha(1a)-adrenergic receptors

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12 December 2020

Movement of retinal along the visual transduction path

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12 December 2020

Analysis of the adrenal angiotensin II receptor with the photoaffinity labeling method

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12 December 2020

Localization of the fourth membrane spanning domain as a ligand binding site in the human platelet alpha 2-adrenergic receptor

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12 December 2020

Identification of amino acid residues of rat angiotensin II receptor for ligand binding by site directed mutagenesis

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12 December 2020

Interaction of glutamine 165 in the fourth transmembrane segment of the human neurokinin-1 receptor with quinuclidine antagonists

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12 December 2020

Electrostatic potential of the acetylcholine binding sites in the nicotinic receptor probed by reactions of binding-site cysteines with charged methanethiosulfonates

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12 December 2020

Identification of peptide binding residues in the extracellular domains of the AT1 receptor

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12 December 2020

Tetrazole and carboxylate groups of angiotensin receptor antagonists bind to the same subsite by different mechanisms

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12 December 2020

Identifiers

DOI

10.1074/JBC.M109.077180

1 reference

28 July 2017

1 reference

28 July 2017

1 reference