The essential role for aromatic cluster in the β3 adrenergic receptor (Q33571267)

28 July 2017

The essential role for aromatic cluster in the β3 adrenergic receptor (English)

1 reference

28 July 2017

Hai-yan Cai

1

1 reference

28 July 2017

Zhi-jian Xu

2

1 reference

28 July 2017

Jie Tang

3

1 reference

28 July 2017

Ying Sun

4

1 reference

28 July 2017

Kai-xian Chen

5

1 reference

28 July 2017

He-yao Wang

6

1 reference

28 July 2017

Wei-liang Zhu

7

1 reference

28 July 2017

language of work or name

1 reference

25 June 2012

1 reference

Acta Pharmacologica Sinica

28 July 2017

1 reference

28 July 2017

33

1 reference

28 July 2017

8

1 reference

28 July 2017

1062-1068

1 reference

https://scigraph.springernature.com/pub.10.1038/aps.2012.55

28 July 2017

0 references

cites work

Structure of a nanobody-stabilized active state of the β(2) adrenoceptor

1 reference

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A conserved aromatic lock for the tryptophan rotameric switch in TM-VI of seven-transmembrane receptors

21 June 2018

1 reference

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The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonist

21 June 2018

1 reference

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Effects of the beta3-adrenoceptor (Adrb3) agonist SR58611A (amibegron) on serotonergic and noradrenergic transmission in the rodent: relevance to its antidepressant/anxiolytic-like profile

21 June 2018

1 reference

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Structure of a beta1-adrenergic G-protein-coupled receptor

21 June 2018

1 reference

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High-resolution crystal structure of an engineered human beta2-adrenergic G protein-coupled receptor

21 June 2018

1 reference

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Location of Trp265 in metarhodopsin II: implications for the activation mechanism of the visual receptor rhodopsin

21 June 2018

1 reference

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Molecular mechanism of 7TM receptor activation--a global toggle switch model

21 June 2018

1 reference

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Structure of bovine rhodopsin in a trigonal crystal form.

21 June 2018

1 reference

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Differential dynamics in the G protein-coupled receptor rhodopsin revealed by solution NMR.

21 June 2018

1 reference

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Beta2 adrenergic receptor activation. Modulation of the proline kink in transmembrane 6 by a rotamer toggle switch

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4011317

Agonist-induced conformational changes in the G-protein-coupling domain of the beta 2 adrenergic receptor

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4011317

Ser203 as well as Ser204 and Ser207 in fifth transmembrane domain of the human beta2-adrenoceptor contributes to agonist binding and receptor activation

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4011317

Mutation of a highly conserved aspartic acid in the beta2 adrenergic receptor: constitutive activation, structural instability, and conformational rearrangement of transmembrane segment 6.

21 June 2018

1 reference

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Species differences in the distribution of beta-adrenoceptor subtypes in bladder smooth muscle

21 June 2018

1 reference

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Agonists induce conformational changes in transmembrane domains III and VI of the beta2 adrenoceptor

21 June 2018

1 reference

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Rhodopsin activation blocked by metal-ion-binding sites linking transmembrane helices C and F.

21 June 2018

1 reference

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Involvement of Asn-293 in stereospecific agonist recognition and in activation of the beta 2-adrenergic receptor

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4011317

Is there a 'lock' for all agonist 'keys' in 7TM receptors?

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4011317

Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins

21 June 2018

1 reference

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Agonist-receptor efficacy. I: Mechanisms of efficacy and receptor promiscuity.

21 June 2018

1 reference

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A single amino acid substitution in the beta-adrenergic receptor promotes partial agonist activity from antagonists

21 June 2018

1 reference

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Molecular characterization of the human beta 3-adrenergic receptor

21 June 2018

1 reference

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Differential transcriptional activation in vitro by NF-kappa B/Rel proteins

21 June 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2012.55

Metal ion site engineering indicates a global toggle switch model for seven-transmembrane receptor activation.

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2012.55

Functional role of the "ionic lock"--an interhelical hydrogen-bond network in family A heptahelical receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2012.55

The retinal conformation and its environment in rhodopsin in light of a new 2.2 A crystal structure

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2012.55

Activation of beta2- and beta3-adrenergic receptors increases brain tryptophan

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2012.55

PROCHECK: a program to check the stereochemical quality of protein structures

21 January 2018

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2012.55

Three-dimensional representations of G protein-coupled receptor structures and mechanisms

21 January 2018

1 reference

12 December 2020

The catecholamine binding site of the beta-adrenergic receptor is formed by juxtaposed membrane-spanning domains

1 reference

12 December 2020

Identification of two serine residues involved in agonist activation of the beta-adrenergic receptor

1 reference

12 December 2020

Fluorescent labeling of purified beta 2 adrenergic receptor. Evidence for ligand-specific conformational changes

1 reference

12 December 2020

Expression and possible functional role of the beta3-adrenoceptor in human and rat detrusor muscle

1 reference

12 December 2020

Insights into the binding modes of human β₃-adrenergic receptor agonists with ligand-based and receptor-based methods

1 reference

12 December 2020

Automated docking using a Lamarckian genetic algorithm and an empirical binding free energy function

1 reference

https://api.crossref.org/works/10.1038%2FAPS.2012.55

7 January 2021

inferred from DOI database lookup

Identifiers

DOI

10.1038/APS.2012.55

1 reference

Dimensions Publication ID

28 July 2017

0 references

1 reference

28 July 2017

1 reference