A conformational switch high-throughput screening assay and allosteric inhibition of the flavivirus NS2B-NS3 protease (Q30145558)

18 October 2017

A conformational switch high-throughput screening assay and allosteric inhibition of the flavivirus NS2B-NS3 protease (English)

1 reference

high-throughput screening

18 October 2017

0 references

author

Matthew Brecher

1

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:28542603%20AND%20SRC:MED&resulttype=core&format=json

11 June 2020

Adham Alifarag

6

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11 June 2020

Laura D Kramer

9

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11 June 2020

Hongmin Li

10

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11 June 2020

author name string

Zhong Li

2

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11 June 2020

Binbin Liu

3

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11 June 2020

Jing Zhang

4

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11 June 2020

Cheri A Koetzner

5

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11 June 2020

Susan A Jones

7

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11 June 2020

Qishan Lin

8

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11 June 2020

language of work or name

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25 May 2017

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18 October 2017

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11 June 2020

volume

13

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11 June 2020

page(s)

e1006411

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11 June 2020

issue

5

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Creative Commons Attribution 4.0 International

11 June 2020

copyright license

start time

25 May 2017

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April 2022 Public Data File from Crossref

copyright status

copyrighted

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cites work

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3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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Towards the design of antiviral inhibitors against flaviviruses: the case for the multifunctional NS3 protein from Dengue virus as a target

3 June 2018

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Mutagenesis of the West Nile virus NS2B cofactor domain reveals two regions essential for protease activity

3 June 2018

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Crystal Structure of the NS3 Protease-Helicase from Dengue Virus

3 June 2018

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3 June 2018

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Structural evidence for regulation and specificity of flaviviral proteases and evolution of theFlaviviridaefold

3 June 2018

1 reference

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Chemical screening methods to identify ligands that promote protein stability, protein crystallization, and structure determination

3 June 2018

1 reference

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Structural basis for the activation of flaviviral NS3 proteases from dengue and West Nile virus.

3 June 2018

1 reference

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Searching for new allosteric sites in enzymes

3 June 2018

1 reference

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Identification of residues in the dengue virus type 2 NS2B cofactor that are critical for NS3 protease activation

3 June 2018

1 reference

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Kinetics of regulated protein-protein interactions revealed with firefly luciferase complementation imaging in cells and living animals

3 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5462475

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3 June 2018

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The structure of unliganded reverse transcriptase from the human immunodeficiency virus type 1

3 June 2018

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Nucleotide sequence of yellow fever virus: implications for flavivirus gene expression and evolution

3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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Crystal structure at 3.5 A resolution of HIV-1 reverse transcriptase complexed with an inhibitor

3 June 2018

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NMR study of complexes between low molecular mass inhibitors and the West Nile virus NS2B-NS3 protease

3 June 2018

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Exploring the binding of peptidic West Nile virus NS2B-NS3 protease inhibitors by NMR.

21 January 2018

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Novel genetically encoded biosensors using firefly luciferase

21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Binding mode of the activity-modulating C-terminal segment of NS2B to NS3 in the dengue virus NS2B-NS3 protease

21 January 2018

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21 January 2018

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10.1371/JOURNAL.PPAT.1006411

21 January 2018

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11 June 2020

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11 June 2020

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