Identification of novel human dipeptidyl peptidase-IV inhibitors of natural origin (part I): virtual screening and activity assays (Q28483681)

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13 February 2020

title

Identification of novel human dipeptidyl peptidase-IV inhibitors of natural origin (part I): virtual screening and activity assays (English)

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13 February 2020

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3

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Adrià Cereto-Massagué

5

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Miquel Mulero

6

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Montserrat Pinent

8

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Anna Ardévol

9

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Santiago Garcia-Vallvé

10

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Gerard Pujadas

11

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1

Laura Guasch

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13 February 2020

author name string

Maria José Ojeda

2

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13 February 2020

Esther Sala

4

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Cristina Valls

7

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13 February 2020

language of work or name

English

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publication date

12 September 2012

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13 February 2020

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volume

7

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issue

9

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13 February 2020

page(s)

e44971

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Creative Commons Attribution 4.0 International

13 February 2020

copyright license

start time

12 September 2012

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April 2022 Public Data File from Crossref

copyright status

copyrighted

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Dipeptidyl-peptidase IV hydrolyses gastric inhibitory polypeptide, glucagon-like peptide-1(7-36)amide, peptide histidine methionine and is responsible for their degradation in human serum

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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27 November 2018

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27 November 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/22984596

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

1-((3S,4S)-4-amino-1-(4-substituted-1,3,5-triazin-2-yl) pyrrolidin-3-yl)-5,5-difluoropiperidin-2-one inhibitors of DPP-4 for the treatment of type 2 diabetes

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22984596

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Sulphostin, a potent inhibitor for dipeptidyl peptidase IV from Streptomyces sp. MK251-43F3

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22984596

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1371/JOURNAL.PONE.0044971

1 reference

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13 February 2020

0 references

1 reference

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13 February 2020

PubMed publication ID

22984596

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22984596%20AND%20SRC:MED&resulttype=core&format=json