Therapeutic potential for novel drugs targeting the type 1 cholecystokinin receptor (Q24628602)

British Journal of Pharmacology

Europe PubMed Central

title

Therapeutic potential for novel drugs targeting the type 1 cholecystokinin receptor (English)

0 references

1 reference

Erin E Cawston

1

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Laurence J Miller

series ordinal

2

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language of work or name

English

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publication date

March 2010

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published in

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volume

159

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issue

5

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page(s)

1009-21

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cites work

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30 May 2018

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30 May 2018

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1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

Advanced qRT-PCR technology allows detection of the cholecystokinin 1 receptor (CCK1R) expression in human pancreas.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

Effect of oral CCK-1 agonist GI181771X on fasting and postprandial gastric functions in healthy volunteers

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

PKC-delta and -epsilon regulate NF-kappaB activation induced by cholecystokinin and TNF-alpha in pancreatic acinar cells

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

Phosphatidylinositide 3-kinase gamma regulates key pathologic responses to cholecystokinin in pancreatic acinar cells

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

Genetic verification of the role of CCK-AR in pancreatic proliferation and blood glucose and insulin regulation using a congenic rat carrying CCK-AR null allele.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

Effect of exogenous cholecystokinin (CCK)-8 on food intake and plasma CCK, leptin, and insulin concentrations in older and young adults: evidence for increased CCK activity as a cause of the anorexia of aging

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

Human pancreatic acinar cells lack functional responses to cholecystokinin and gastrin

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

Loxiglumide, a CCK-A receptor antagonist, stimulates calorie intake and hunger feelings in humans

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

SR146131: a new potent, orally active, and selective nonpeptide cholecystokinin subtype 1 receptor agonist. II. In vivo pharmacological characterization.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

Adenovirus-mediated gene transfer of RasN17 inhibits specific CCK actions on pancreatic acinar cells.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

Early NF-kappaB activation is associated with hormone-induced pancreatitis.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

Endogenous cholecystokinin in postprandial lower esophageal sphincter function and fundic tone in humans.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

CCK in anxiety and cognitive processes.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

Cyclic ADP-ribose as an endogenous regulator of the non-skeletal type ryanodine receptor Ca2+ channel.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

Characterization of cholecystokinin receptors on the human gallbladder.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

Structure-activity relationship studies on cholecystokinin: analogues with partial agonist activity

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

A71378: a CCK agonist with high potency and selectivity for CCK-A receptors.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2839260

Multiple sources of 1,2-diacylglycerol in isolated rat pancreatic acini stimulated by cholecystokinin. Involvement of phosphatidylinositol bisphosphate and phosphatidylcholine hydrolysis

28 November 2018

1 reference

12 December 2020

Physiological plasma concentrations of cholecystokinin stimulate pancreatic enzyme secretion and gallbladder contraction in man

1 reference

12 December 2020

Pharmacological dissociation of responses to CCK and gastric loads in rat mechanosensitive vagal afferents

1 reference

12 December 2020

Cholecystokinin rapidly activates mitogen-activated protein kinase in rat pancreatic acini

1 reference

12 December 2020

Two functionally distinct cholecystokinin receptors show different modes of action on Ca2+ mobilization and phospholipid hydrolysis in isolated rat pancreatic acini. Studies using a new cholecystokinin analog, JMV-180

1 reference

12 December 2020

Analogs of CCK incorporating conformationally constrained replacements for Asp32

1 reference

12 December 2020

Transport of cholecystokinin (CCK) binding sites in subdiaphragmatic vagal branches

1 reference

12 December 2020

Receptor-activated cytoplasmic Ca2+ spiking mediated by inositol trisphosphate is due to Ca2(+)-induced Ca2+ release

1 reference

12 December 2020

Effects of three different cholecystokinin receptor antagonists on basal and stimulated insulin and glucagon secretion in mice

1 reference

12 December 2020

High-affinity CCK-A receptors on the vagus nerve mediate CCK-stimulated pancreatic secretion in rats

1 reference

12 December 2020

Regulation of protein synthesis by cholecystokinin in rat pancreatic acini involves PHAS-I and the p70 S6 kinase pathway

1 reference

12 December 2020

Bioactivity of cholecystokinin analogues: CCK-8 is not more potent than CCK-33

1 reference

12 December 2020

A cloned CCK-A receptor transduces multiple signals in response to full and partial agonists

1 reference

12 December 2020

Calcium release by cholecystokinin analogue OPE is IP3 dependent in single rat pancreatic acinar cells

1 reference

12 December 2020

Pancreas growth, tyrosine kinase, PtdIns 3-kinase, and PLD involve high-affinity CCK-receptor occupation

1 reference

12 December 2020

Chemokine gene expression in rat pancreatic acinar cells is an early event associated with acute pancreatitis

1 reference

12 December 2020

Effect of dexloxiglumide and spiroglumide, two new CCK-receptor antagonists, on gastric emptying and secretion in the rat: evaluation of their receptor selectivity in vivo

1 reference

12 December 2020

CCK satiety is differentially mediated by high- and low-affinity CCK receptors in mice and rats

1 reference

12 December 2020

Structure of porcine cholecystokinin-pancreozymin. 1. Cleavage with thrombin and with trypsin

1 reference

12 December 2020

Pancreozymin, a stimulant of the secretion of pancreatic enzymes in extracts of the small intestine

1 reference

12 December 2020

Complex role of protein kinase C in mediating the supramaximal inhibition of pancreatic secretion observed with cholecystokinin

1 reference

12 December 2020

1 reference

12 December 2020

beta-Adrenergic receptor kinase. Activity of partial agonists for stimulation of adenylate cyclase correlates with ability to promote receptor phosphorylation

1 reference

12 December 2020

Promiscuous Coupling of Receptors to Gq Class α Subunits and Effector Proteins in Pancreatic and Submandibular Gland Cells

1 reference

12 December 2020

Binding of cholecystokinin to high affinity receptors on isolated rat pancreatic acini

1 reference

12 December 2020

NF-kappaB/Rel activation in cerulein pancreatitis

1 reference

12 December 2020

CCK receptor dysfunction in muscle membranes from human gallbladders with cholesterol stones

1 reference

12 December 2020

Jun kinases are rapidly activated by cholecystokinin in rat pancreas both in vitro and in vivo

1 reference

12 December 2020

Stimulation of both CCK-A and CCK-B receptors activates MAP kinases in AR42J and receptor-transfected CHO cells

1 reference

12 December 2020

The design and synthesis of the high efficacy, non-peptide CCK 1 receptor agonist PD 170292

1 reference

12 December 2020

CCK activates p90rsk in rat pancreatic acini through protein kinase C

1 reference

12 December 2020

Structure activity of C-terminal modified analogs of Ac-CCK-7

1 reference

12 December 2020

Intracellular glucose switches between cyclic ADP-ribose and inositol trisphosphate triggering of cytosolic Ca2+ spiking

1 reference

12 December 2020

Characterization of novel peptoid agonists for the CCK-A receptor

1 reference

12 December 2020

Plasma cholecystokinin and pancreatic polypeptide secretion in response to bombesin, meal ingestion and modified sham feeding in lean and obese persons

1 reference

12 December 2020

A major quantitative trait locus co-localizing with cholecystokinin type A receptor gene influences poor pancreatic proliferation in a spontaneously diabetogenic rat

1 reference

12 December 2020

The New Biology of Gastrointestinal Hormones

1 reference

12 December 2020

The interaction of caerulein with the rat pancreas. 1. Specific binding of [3H]caerulein on plasma membranes and evidence for negative cooperativity

1 reference

12 December 2020

Synthesis and biological evaluation of potent, selective, hexapeptide CCK-A agonist anorectic agents

1 reference

12 December 2020

High-affinity CCK receptors are coupled to phospholipase A2 pathways to mediate pancreatic amylase secretion

1 reference

12 December 2020

Affinity and intrinsic-activity in the theory of competitive inhibition. III. Homologous decamethonium-derivatives and succinyl-choline-esters

1 reference

12 December 2020