The discovery of Polo-like kinase 4 inhibitors: identification of (1R,2S).2-(3-((E).4-(((cis).2,6-dimethylmorpholino)methyl)styryl). 1H.indazol-6-yl)-5 '-methoxyspiro[cyclopropane-1,3 '-indolin]-2 '-one (CFI-400945) as a potent, orally active antitu (Q95784946)
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scientific article published in January 2015
Language | Label | Description | Also known as |
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English | The discovery of Polo-like kinase 4 inhibitors: identification of (1R,2S).2-(3-((E).4-(((cis).2,6-dimethylmorpholino)methyl)styryl). 1H.indazol-6-yl)-5 '-methoxyspiro[cyclopropane-1,3 '-indolin]-2 '-one (CFI-400945) as a potent, orally active antitu |
scientific article published in January 2015 |
Statements
The discovery of Polo-like kinase 4 inhibitors: identification of (1R,2S).2-(3-((E).4-(((cis).2,6-dimethylmorpholino)methyl)styryl). 1H.indazol-6-yl)-5'-methoxyspiro[cyclopropane-1,3'-indolin]-2'-one (CFI-400945) as a potent, orally active antitumor agent (English)
Peter B Sampson
Yong Liu
Bryan Forrest
Graham Cumming
Sze-Wan Li
Narendra Kumar Patel
Louise Edwards
Radoslaw Laufer
Miklos Feher
Fuqiang Ban
Donald E Awrey
Guodong Mao
Olga Plotnikova
Jacqueline M Mason
Xunyi Luo
Vincent Nadeem
Xin Wei
Reza Kiarash
Brian Madeira
Ping Huang
Tak W Mak
Guohua Pan