Virtual Screening for Selective Allosteric mGluR1 Antagonists and Structure–Activity Relationship Investigations for Coumarine Derivatives (Q60722382)

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7 January 2020

title

Virtual screening for selective allosteric mGluR1 antagonists and structure-activity relationship investigations for coumarine derivatives (English)

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Christopher G. Parsons

10

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Tanja Weil

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Gisbert Schneider

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author name string

Tobias Noeske

1

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Aigars Jirgensons

2

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Igors Starchenkovs

3

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Steffen Renner

4

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Ieva Jaunzeme

5

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Dina Trifanova

6

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Mirko Hechenberger

7

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Tanja Bauer

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Valerjans Kauss

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publication date

1 December 2007

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volume

2

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issue

12

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page(s)

1763-1773

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Molecular basis of receptor/G-protein-coupling selectivity

7 January 2020

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Mutational analysis of muscarinic acetylcholine receptors: structural basis of ligand/receptor/G protein interactions

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G protein-mediated inhibition of phosphoinositide metabolism evoked by metabotropic glutamate receptors in frog oocytes

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Metabotropic glutamate receptors: a new target for the therapy of neurodegenerative disorders?

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1-Aminoindan-1,5-dicarboxylic acid and (S)-(+)-2-(3'-carboxybicyclo[1.1.1] pentyl)-glycine, two mGlu1 receptor-preferring antagonists, reduce neuronal death in in vitro and in vivo models of cerebral ischaemia

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Metabotropic glutamate receptor mRNA expression in rat spinal cord.

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Evidence for a role of metabotropic glutamate receptors in sustained nociceptive inputs to rat dorsal horn neurons

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Allosteric modulators of group I metabotropic glutamate receptors: novel subtype-selective ligands and therapeutic perspectives.

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The non-competitive antagonists 2-methyl-6-(phenylethynyl)pyridine and 7-hydroxyiminocyclopropan[b]chromen-1a-carboxylic acid ethyl ester interact with overlapping binding pockets in the transmembrane region of group I metabotropic glutamate recepto

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Synthesis, structure-activity relationship, and receptor pharmacology of a new series of quinoline derivatives acting as selective, noncompetitive mGlu1 antagonists

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7 January 2021

Mutational analysis and molecular modeling of the allosteric binding site of a novel, selective, noncompetitive antagonist of the metabotropic glutamate 1 receptor

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7 January 2021

Group I metabotropic glutamate receptors: implications for brain diseases

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Insight into the function of Group I and Group II metabotropic glutamate (mGlu) receptors: behavioural characterization and implications for the treatment of CNS disorders

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Virtual screening and fast automated docking methods.

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Molecular modeling of the mGluR1 metabotropic glutamate receptor transmembrane domain and construction of the model of its dimer.

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Pharmacological and biochemical actions of simple coumarins: natural products with therapeutic potential

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The Vapor Phase Rearrangement of Thioncarbonates and Thioncarbamates

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7 January 2021

The Conversion of Phenols to Thiophenols via Dialkylthiocarbamates1

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Crystal structure of rhodopsin: A G protein-coupled receptor

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Mutational Analysis and Molecular Modeling of the Binding Pocket of the Metabotropic Glutamate 5 Receptor Negative Modulator 2-Methyl-6-(phenylethynyl)-pyridine

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7 January 2021

Identifiers

DOI

10.1002/CMDC.200700151

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7 January 2020

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