Structure–activity studies on nociceptin/orphanin FQ: from full agonist, to partial agonist, to pure antagonist (Q57951324)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10668183%20AND%20SRC:MED&resulttype=core&format=json

3 November 2019

title

Structure-activity studies on nociceptin/orphanin FQ: from full agonist, to partial agonist, to pure antagonist (English)

1 reference

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3 November 2019

0 references

1

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3 November 2019

Remo Guerrini

series ordinal

2

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3 November 2019

author name string

G Calo

series ordinal

3

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3 November 2019

D Regoli

series ordinal

4

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3 November 2019

publication date

1 November 1999

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3 November 2019

1 reference

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3 November 2019

volume

54

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3 November 2019

issue

11-12

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3 November 2019

page(s)

810-825

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Molecular cloning and tissue distribution of a putative member of the rat opioid receptor gene family that is not a mu, delta or kappa opioid receptor type

3 November 2019

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Nociceptin/orphanin FQ microinjected into hippocampus impairs spatial learning in rats.

7 January 2021

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Facilitation of long-term potentiation and memory in mice lacking nociceptin receptors.

7 January 2021

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Injections of nociceptin into nucleus accumbens shell or ventromedial hypothalamic nucleus increase food intake.

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Orphanin FQ stimulates prolactin and growth hormone release in male and female rats.

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Inhibition of rat oxytocin and vasopressin supraoptic nucleus neurons by nociceptin in vitro.

7 January 2021

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Determination of activity for nociceptin in the mouse vas deferens

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Naloxone-insensitive inhibition of acetylcholine release from parasympathetic nerves innervating guinea-pig trachea by the novel opioid, nociceptin

7 January 2021

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Inhibition of tachykinin release from peripheral endings of sensory nerves by nociceptin, a novel opioid peptide

7 January 2021

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Prejunctional modulation by nociceptin of nerve-mediated inotropic responses in guinea-pig left atrium

7 January 2021

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Inhibition by nociceptin of neurogenic inflammation and the release of SP and CGRP from sensory nerve terminals

7 January 2021

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Effect of nociceptin on heart rate and blood pressure in anaesthetized rats.

7 January 2021

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The inhibitory effect of nociceptin on the micturition reflex in anaesthetized rats

7 January 2021

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Structure, tissue distribution, and chromosomal localization of the prepronociceptin gene

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Nocistatin, a peptide that blocks nociceptin action in pain transmission

7 January 2021

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Estimated conformation, orientation, and accumulation of dynorphin A-(1-13)-tridecapeptide on the surface of neutral lipid membranes.

7 January 2021

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Structures that delineate orphanin FQ and dynorphin A pharmacological selectivities

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Different domains of the ORL1 and kappa-opioid receptors are involved in recognition of nociceptin and dynorphin A.

7 January 2021

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Molecular modelling of the ORL1 receptor and its complex with nociceptin

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Nociceptin receptor activation inhibits tachykinergic non adrenergic non cholinergic contraction of guinea pig isolated bronchus.

7 January 2021

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7 January 2021

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Nociceptin receptor coupling to a potassium conductance in rat locus coeruleus neurones in vitro

7 January 2021

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The effect of nociceptin on Ca2+ channel current and intracellular Ca2+ in the SH-SY5Y human neuroblastoma cell line

7 January 2021

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7 January 2021

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Association of aminopeptidase N and endopeptidase 24.15 inhibitors potentiate behavioral effects mediated by nociceptin/orphanin FQ in mice

7 January 2021

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In vivo metabolism of nociceptin/orphanin FQ in rat hippocampus.

7 January 2021

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Biotransformation of nociceptin/orphanin FQ by enzyme activity from morphine-naive and morphine-treated cell cultures.

7 January 2021

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7 January 2021

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Pharmacological characterization of the nociceptin receptor mediating hyperalgesia in the mouse tail withdrawal assay

7 January 2021

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Cardiovascular effects of nociceptin in unanesthetized mice

7 January 2021

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7 January 2021

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Identifiers

DOI

10.1016/S0014-827X(99)00108-1

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3 November 2019

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