Characterization of a novel 5-HT4 receptor antagonist of the azabicycloalkyl benzimidazolone class: DAU 6285 (Q48523967)

12 February 2018

title

Characterization of a novel 5-HT4 receptor antagonist of the azabicycloalkyl benzimidazolone class: DAU 6285 (English)

1 reference

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heterocyclic bridged bicyclo compounds

13 September 2022

main subject

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13 September 2022

Serotonin antagonists

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6 December 2023

author name string

A. Dumuis

1

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13 September 2022

H. Gozlan

2

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13 September 2022

M. Sebben

3

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13 September 2022

H. Ansanay

4

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13 September 2022

C. A. Rizzi

5

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13 September 2022

M. Turconi

6

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13 September 2022

E. Monferini

7

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13 September 2022

E. Giraldo

8

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13 September 2022

P. Schiantarelli

9

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13 September 2022

H. Ladinsky

10

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13 September 2022

language of work or name

English

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National Center for Biotechnology Information

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=1320204

13 September 2022

publication date

1 March 1992

1 reference

12 February 2018

full work available at URL

http://link.springer.com/article/10.1007/BF00168685/fulltext.html

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https://api.crossref.org/works/10.1007/BF00168685

http://link.springer.com/content/pdf/10.1007/BF00168685.pdf

6 December 2023

file format

Portable Document Format

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https://api.crossref.org/works/10.1007/BF00168685

http://link.springer.com/content/pdf/10.1007/BF00168685

6 December 2023

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Naunyn-Schmiedeberg's Archives of Pharmacology

6 December 2023

published in

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12 February 2018

volume

345

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12 February 2018

issue

3

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12 February 2018

page(s)

264-269

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12 February 2018

https://scigraph.springernature.com/pub.10.1007/bf00168685

exact match

0 references

cites work

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12 December 2020

BRL 24924: a potent agonist at a non-classical 5-HT receptor positively coupled with adenylate cyclase in colliculi neurons

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Binding characteristics of 3H-prazosin to rat brain α-adrenergic receptors

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Synthesis of a new class of 2,3-dihydro-2-oxo-1H-benzimidazole-1-carboxylic acid derivatives as highly potent 5-HT3 receptor antagonists

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The gastrointestinal prokinetic benzamide derivatives are agonists at the non-classical 5-HT receptor (5-HT4) positively coupled to adenylate cyclase in neurons

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12 December 2020

Activation of a myenteric 5-hydroxytryptamine-like receptor by metoclopramide

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12 December 2020

A 5-HT receptor in the central nervous system, positively coupled with adenylate cyclase, is antagonized by ICS 205 930.

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12 December 2020

SDZ 205–557, a selective antagonist at 5-HT4 receptors in the isolated guinea pig ileum

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12 December 2020

Some quantitative uses of drug antagonists

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12 December 2020

Mediation of 5-hydroxytryptamine-induced tachycardia in the pig by the putative 5-HT4 receptor

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12 December 2020

MDL 72222: a potent and highly selective antagonist at neuronal 5-hydroxytryptamine receptors.

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12 December 2020

Alpha-noradrenergic receptor binding in mammalian brain: Differential labeling of agonist and antagonist states

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12 December 2020

Dopamine receptor binding: Differentiation of agonist and antagonist states with 3H-dopamine and 3H-haloperidol

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12 December 2020

Characterization of the binding of 3H-SCH 23390, a selective D-1 receptor antagonist ligand, in rat striatum.

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12 December 2020

Aging associated changes in serotoninergic and dopaminergic pre- and postsynaptic neurochemical markers in the rat brain

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12 December 2020

Pharmacological characterization of a neuronal receptor for 5-hydroxytryptamine in guinea pig ileum with properties similar to the 5-hydroxytryptamine receptor.

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12 December 2020

Novel enteric 5-HT4 receptors and gastrointestinal prokinetic action

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12 December 2020

Increased gut cholinergic activity and antagonism of 5-hydroxytryptamine M-receptors by BRL 24924: potential clinical importance of BRL 24924.

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12 December 2020

5-HT1D receptors in guinea-pig and pigeon brain. Radioligand binding and biochemical studies

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A 5-hydroxytryptamine receptor in human atrium

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12 December 2020

The 5-HT4 receptor: naughty, but nice

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12 December 2020

Synaptogenesis of cultured striatal neurons in serum-free medium: a morphological and biochemical study

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12 December 2020

Study of the contractile effect of 5-hydroxytryptamine (5-HT) in the isolated longitudinal muscle strip from guinea-pig ileum. Evidence for two distinct release mechanisms.

1 reference

12 December 2020

Further characterization, by use of tryptamine and benzamide derivatives, of the putative 5-HT4 receptor mediating tachycardia in the pig

1 reference

12 December 2020

Identification of putative 5-HT4 receptors in guinea-pig ascending colon

1 reference

12 December 2020

Azabicycloalkyl benzimidazolone derivatives as a novel class of potent agonists at the 5-HT4 receptor positively coupled to adenylate cyclase in braina

1 reference

12 December 2020

Pharmacological characterization of 5-hydroxytryptamine4(5-HT4) receptors positively coupled to adenylate cyclase in adult guinea pig hippocampal membranes: effect of substituted benzamide derivatives.

1 reference

12 December 2020

SDZ 205-557, a selective, surmountable antagonist for 5-HT4 receptors in the isolated guinea pig ileum

1 reference

12 December 2020

Pharmacological properties of a novel class of 5-HT3 receptor antagonists

1 reference

12 December 2020

Identification of serotonin M-receptor subtypes and their specific blockade by a new class of drugs.

1 reference

12 December 2020

Zacopride, a potent 5-HT3 antagonist

1 reference

12 December 2020

Binding profile of a novel cardioselective muscarine receptor antagonist, AF-DX 116, to membranes of peripheral tissues and brain in the rat.

1 reference

12 December 2020

5-Methoxytryptamine and 2-methyl-5-hydroxytryptamine-induced desensitization as a discriminative tool for the 5-HT3 and putative 5-HT4 receptors in guinea pig ileum

1 reference

12 December 2020

5-Hydroxytryptamine4 receptors mediate relaxation of the rat oesophageal tunica muscularis mucosae

1 reference

12 December 2020

Investigation into the 5-hydroxytryptamine receptor mediating smooth muscle relaxation in the rat oesophagus

1 reference

12 December 2020

Piglet sinoatrial 5-HT receptors resemble human atrial 5-HT4-like receptors

1 reference

12 December 2020

Common pharmacological and physico-chemical properties of 5-HT3 binding sites in the rat cerebral cortex and NG 108-15 clonal cells.

1 reference

12 December 2020

Identifiers

DOI

10.1007/BF00168685

1 reference

12 February 2018

1 reference

12 February 2018