Calcimimetic and calcilytic therapies for inherited disorders of the calcium-sensing receptor signalling pathway. (Q47414200)

15 January 2018

title

Calcimimetic and calcilytic therapies for inherited disorders of the calcium-sensing receptor signalling pathway. (English)

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15 January 2018

author

Fadil M. Hannan

series ordinal

1

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15 January 2018

Rajesh Thakker

series ordinal

3

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15 January 2018

Mie K Olesen

object named as

Mie K Olesen

series ordinal

2

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language of work or name

English

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publication date

11 November 2017

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15 January 2018

British Journal of Pharmacology

published in

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15 January 2018

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: G protein-coupled receptors

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Positive and negative allosteric modulators of the Ca2+-sensing receptor interact within overlapping but not identical binding sites in the transmembrane domain

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21 January 2018

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PubMed Central

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6177618

Recurrent pancreatitis in a patient with familial hypocalciuric hypercalcaemia treated successfully with cinacalcet

2 November 2018

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PubMed Central

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6177618

Calcilytic compounds: potent and selective Ca2+ receptor antagonists that stimulate secretion of parathyroid hormone.

2 November 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=6177618

The effects of ronacaleret, a calcium-sensing receptor antagonist, on bone mineral density and biochemical markers of bone turnover in postmenopausal women with low bone mineral density

2 November 2018

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12 December 2020

Short-term inhibition of parathyroid hormone secretion by a calcium-receptor agonist in patients with primary hyperparathyroidism

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12 December 2020

Agonist-driven maturation and plasma membrane insertion of calcium-sensing receptors dynamically control signal amplitude

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12 December 2020

Novel activating mutations of the calcium-sensing receptor: the calcilytic NPS-2143 mitigates excessive signal transduction of mutant receptors

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12 December 2020

An orally active calcium-sensing receptor antagonist that transiently increases plasma concentrations of PTH and stimulates bone formation

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12 December 2020

Correction of hypercalcaemia by cinacalcet in familial hypocalciuric hypercalcaemia

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12 December 2020

Cinacalcet Treatment in an Adolescent With Concurrent 22q11.2 Deletion Syndrome and Familial Hypocalciuric Hypercalcemia Type 3 Caused by AP2S1 Mutation

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12 December 2020

A calcimimetic agent acutely suppresses parathyroid hormone levels in patients with chronic renal failure. Rapid communication

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12 December 2020

Identifiers

DOI

10.1111/BPH.14086

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15 January 2018

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15 January 2018