Asymmetric synthesis of propargylamines as amino acid surrogates in peptidomimetics. (Q47155287)

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7 April 2020

title

Asymmetric synthesis of propargylamines as amino acid surrogates in peptidomimetics (English)

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7 April 2020

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7 April 2020

Matthias Wünsch

1

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7 April 2020

David Schröder

2

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7 April 2020

Nils Janson

6

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7 April 2020

Jasmin Simon

8

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7 April 2020

Shari Heidemeyer

9

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7 April 2020

Alessa Hinzmann

13

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7 April 2020

Hans-Georg Stammler

15

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7 April 2020

author name string

Tanja Fröhr

3

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7 April 2020

Lisa Teichmann

4

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7 April 2020

Sebastian Hedwig

5

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7 April 2020

Clara Belu

7

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Philipp Holtkamp

10

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7 April 2020

Jens Rudlof

11

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7 April 2020

Lennard Klemme

12

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7 April 2020

Beate Neumann

14

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7 April 2020

publication date

15 November 2017

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Beilstein Journal of Organic Chemistry

7 April 2020

published in

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volume

13

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7 April 2020

page(s)

2428-2441

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Phenylalanine and Phenylglycine Analogues as Arginine Mimetics in Dengue Protease Inhibitors

7 April 2020

cites work

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Applications of Fluorine in Medicinal Chemistry

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Selectivity of commonly used pharmacological inhibitors for cystathionine β synthase (CBS) and cystathionine γ lyase (CSE).

23 May 2018

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Microwave-assisted solvent-free synthesis of enantiomerically pure N-(tert-butylsulfinyl)imines

23 May 2018

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Universal peptidomimetics.

23 May 2018

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23 May 2018

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Functional studies of Plasmodium falciparum dipeptidyl aminopeptidase I using small molecule inhibitors and active site probes

23 May 2018

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23 May 2018

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Synthesis and applications of tert-butanesulfinamide

23 May 2018

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The tert-butylsulfinamide lynchpin in transition-metal-mediated multiscaffold library synthesis

23 May 2018

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"Clicktophycin-52": a bioactive cryptophycin-52 triazole analogue

23 May 2018

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Nonpeptidic Tetrafluorophenoxymethyl Ketone Cruzain Inhibitors as Promising New Leads for Chagas Disease Chemotherapy

23 May 2018

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Efavirenz: a decade of clinical experience in the treatment of HIV.

23 May 2018

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Another ten stories in antiviral drug discovery (part C): "Old" and "new" antivirals, strategies, and perspectives

23 May 2018

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23 May 2018

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The role of fluorine in medicinal chemistry

23 May 2018

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23 May 2018

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Characterization and optimization of selective, nonpeptidic inhibitors of cathepsin S with an unprecedented binding mode

23 May 2018

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Are all antidepressants really the same? The case of fluoxetine: a systematic review.

23 May 2018

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Olanzapine/fluoxetine combination for bipolar depression and other mood disorders: a review

23 May 2018

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23 May 2018

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23 May 2018

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Influence of HMPA on the stereochemical outcome of the addition of a racemic allenylzinc onto enantiopure N-tert-butanesulfinimines: stereoselective access to enantiopure cis-ethynylaziridines.

23 May 2018

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The chemistry of trifluoromethyl imines and related acetals derived from fluoral

23 May 2018

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New antivirals and antiviral resistance.

23 May 2018

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Activity and properties of para-aminobenzyl penicillin.

23 May 2018

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Role of fluoxetine in anorexia nervosa

23 May 2018

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N-tert-Butanesulfinyl Imines: Versatile Intermediates for the Asymmetric Synthesis of Amines

23 May 2018

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23 May 2018

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15 August 2018

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15 August 2018

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15 August 2018

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The total synthesis of tubulysin D.

15 August 2018

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15 August 2018

1 reference

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15 August 2018

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15 August 2018

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15 August 2018

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15 August 2018

1 reference

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1 reference

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29 September 2018

1 reference

12 December 2020

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1 reference

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Synthesis and reactivity of mixed alkynylalanes by direct triethylamine-catalyzed alumination of terminal alkynes

1 reference

12 December 2020

Asymmetric syntheses of 1-aryl-2,2,2-trifluoroethylamines via diastereoselective 1,2-addition of arylmetals to 2-methyl-N-(2,2,2-trifluoroethylidene)propane-2-sulfinamide

1 reference

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Diastereoselective alkynylation of N-p-tolylsulfinylimines with aluminum acetylides

1 reference

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Highly diastereoselective addition of alkynylmagnesium chlorides to N-tert-butanesulfinyl aldimines: a practical and general access to chiral alpha-branched amines

1 reference

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Predicting the activity of antimicrobial peptides with amino acid topological information

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A general and regioselective synthesis of 5-trifluoromethyl-pyrazoles

1 reference

12 December 2020

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1 reference

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1 reference

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1 reference

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Identifiers

DOI

10.3762/BJOC.13.240

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29234470%20AND%20SRC:MED&resulttype=core&format=json

7 April 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29234470%20AND%20SRC:MED&resulttype=core&format=json

7 April 2020

PubMed publication ID

29234470

1 reference