Rational Design of Selective Allosteric Inhibitors of PHGDH and Serine Synthesis with Anti-tumor Activity. (Q46438080)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:28042046%20AND%20SRC:MED&resulttype=core&format=json

4 April 2020

title

Rational Design of Selective Allosteric Inhibitors of PHGDH and Serine Synthesis with Anti-tumor Activity (English)

1 reference

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4 April 2020

1 reference

6

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4 April 2020

Maria V Liberti

2

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4 April 2020

author name string

Qian Wang

1

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4 April 2020

Pei Liu

3

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4 April 2020

Xiaobing Deng

4

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4 April 2020

Ying Liu

5

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4 April 2020

Luhua Lai

7

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publication date

29 December 2016

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4 April 2020

published in

Cell chemical biology

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volume

24

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issue

1

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4 April 2020

page(s)

55-65

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Motions of Allosteric and Orthosteric Ligand-Binding Sites in Proteins are Highly Correlated

4 April 2020

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Phosphoglycerate dehydrogenase is dispensable for breast tumor maintenance and growth

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10 July 2018

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10 July 2018

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10 July 2018

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10 July 2018

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10 July 2018

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10 July 2018

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10 July 2018

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10 July 2018

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10 July 2018

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10 July 2018

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10 July 2018

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10 July 2018

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Validating and enabling phosphoglycerate dehydrogenase (PHGDH) as a target for fragment-based drug discovery in PHGDH-amplified breast cancer.

10 July 2018

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15 August 2018

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15 August 2018

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15 August 2018

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15 August 2018

Identifiers

DOI

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