Fluorine substitution can block CYP3A4 metabolism-dependent inhibition: identification of (S)-N-[1-(4-fluoro-3- morpholin-4-ylphenyl)ethyl]-3- (4-fluorophenyl)acrylamide as an orally bioavailable KCNQ2 opener devoid of CYP3A4 metabolism-dependent in (Q44557212)

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scientific article published in August 2003
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English
Fluorine substitution can block CYP3A4 metabolism-dependent inhibition: identification of (S)-N-[1-(4-fluoro-3- morpholin-4-ylphenyl)ethyl]-3- (4-fluorophenyl)acrylamide as an orally bioavailable KCNQ2 opener devoid of CYP3A4 metabolism-dependent in
scientific article published in August 2003

    Statements

    Fluorine substitution can block CYP3A4 metabolism-dependent inhibition: identification of (S)-N-[1-(4-fluoro-3- morpholin-4-ylphenyl)ethyl]-3- (4-fluorophenyl)acrylamide as an orally bioavailable KCNQ2 opener devoid of CYP3A4 metabolism-dependent in (English)
    Yong-Jin Wu
    Carl D Davis
    Steven Dworetzky
    William C Fitzpatrick
    David Harden
    Ronald J Knox
    Amy E Newton
    Thomas Philip
    Craig Polson
    Digavalli V Sivarao
    Li-Qiang Sun
    Svetlana Tertyshnikova
    David Weaver
    Suresh Yeola
    Mary Zoeckler
    Michael W Sinz
    1 August 2003
    3778-3781

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