Transition-state characterization: a new approach combining inhibitor analogs and variation in enzyme structure (Q44502461)

reason for preferred rank

3 December 2017

Transition-state characterization: a new approach combining inhibitor analogs and variation in enzyme structure (English)

1 reference

11 November 2022

Transition-state characterization: a new approach combining inhibitor analogues and variation in enzyme structure (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1734971

11 November 2022

1 reference

11 November 2022

3

Rutter WJ

1 reference

3 December 2017

M. A. Phillips

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1734971

11 November 2022

A. P. Kaplan

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1734971

11 November 2022

P. A. Bartlett

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1734971

11 November 2022

language of work or name

English

0 references

publication date

1 February 1992

1 reference

3 December 2017

4 February 1992

1 reference

National Center for Biotechnology Information

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=1734971

full work available at URL

11 November 2022

number of pages

5

1 reference

based on heuristic

inferred from page(s)

https://pubs.acs.org/doi/pdf/10.1021/bi00119a003

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11 November 2022

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3 December 2017

31

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3 December 2017

4

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3 December 2017

959-963

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Phosphonamidates as transition-state analogue inhibitors of thermolysin.

3 December 2017

2

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Possible role for water dissociation in the slow binding of phosphorus-containing transition-state-analogue inhibitors of thermolysin

11 November 2022

3

1 reference

Diffusion-limited component of reactions catalyzed by Bacillus cereus beta-lactamase I.

11 November 2022

4

1 reference

6 Statistical analysis of enzyme kinetic data

11 November 2022

7

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Analytical molecular surface calculation

11 November 2022

8

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Solvent-accessible surfaces of proteins and nucleic acids

11 November 2022

9

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Reversible inhibitors of beta-glucosidase

11 November 2022

10

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Adenosine deaminase and adenylate deaminase: comparative kinetic studies with transition state and ground state analogue inhibitors

11 November 2022

11

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Inhibition of carboxypeptidase A by ketones and alcohols that are isosteric with peptide substrates

11 November 2022

12

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Phosphonate analogues of carboxypeptidase A substrates are potent transition-state analogue inhibitors

11 November 2022

13

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A linear equation that describes the steady-state kinetics of enzymes and subcellular particles interacting with tightly bound inhibitors

11 November 2022

14

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Evidence against a crucial role for the phenolic hydroxyl of Tyr-248 in peptide and ester hydrolyses catalyzed by carboxypeptidase A: comparative studies of the pH dependencies of the native and Phe-248-mutant forms

11 November 2022

15

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Synthesis and evaluation of an inhibitor of carboxypeptidase A with a Ki value in the femtomolar range

11 November 2022

17

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(Phosphinyloxy)acyl amino acid inhibitors of angiotensin converting enzyme (ACE). 1. Discovery of (S)-1-[6-amino-2-[[hydroxy(4-phenylbutyl)phosphinyl]oxy]-1-oxohexyl]-L -proline a novel orally active inhibitor of ACE.

11 November 2022

18

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Crystal structure of the complex of carboxypeptidase A with a strongly bound phosphonate in a new crystalline form: comparison with structures of other complexes

11 November 2022

19

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Comparison of the structures of three carboxypeptidase A-phosphonate complexes determined by X-ray crystallography

11 November 2022

20

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Enzymatic Catalysis and Transition-State Theory

11 November 2022

22

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Transition-state analogues in protein crystallography: probes of the structural source of enzyme catalysis

11 November 2022

23

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Ketone-substrate analogues of Clostridium histolyticum collagenases: tight-binding transition-state analogue inhibitors

11 November 2022

25

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Molecular Architecture and Biological Reactions

11 November 2022

26

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Use of peptide aldehydes to generate transition-state analogs of elastase

11 November 2022

31

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Phosphorus-containing inhibitors of angiotensin-converting enzyme

11 November 2022

32

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Direct Brønsted analysis of the restoration of activity to a mutant enzyme by exogenous amines

11 November 2022

33

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Transition state analog inhibitors and enzyme catalysis

11 November 2022

34

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11 November 2022

Identifiers

DOI

10.1021/BI00119A003

1 reference

3 December 2017

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