Influence of imidazole replacement in different structural classes of histamine H(3)-receptor antagonists (Q43625285)

25 November 2017

Influence of imidazole replacement in different structural classes of histamine H(3)-receptor antagonists (English)

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25 November 2017

Meier G

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25 November 2017

Apelt J

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25 November 2017

Reichert U

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25 November 2017

Grassmann S

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25 November 2017

Ligneau X

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25 November 2017

Elz S

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25 November 2017

Leurquin F

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25 November 2017

Ganellin CR

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25 November 2017

Schwartz JC

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25 November 2017

Schunack W

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25 November 2017

Stark H

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25 November 2017

language of work or name

English

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publication date

1 June 2001

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European Journal of Pharmaceutical Sciences

25 November 2017

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25 November 2017

13

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25 November 2017

249-259

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25 November 2017

3

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Design, synthesis, and structure-activity relationships of acetylene-based histamine H3 receptor antagonists.

25 November 2017

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

[3H]-thioperamide as a radioligand for the histamine H3 receptor in rat cerebral cortex

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https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Autoregulation of histamine release in brain by presynaptic H3-receptors

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https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Autoinhibition of histamine synthesis mediated by presynaptic H3-receptors

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7 January 2021

Highly potent and selective ligands for histamine H3-receptors

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https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Inhibition of cortical acetylcholine release and cognitive performance by histamine H3 receptor activation in rats

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7 January 2021

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

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https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Synthesis and histamine H3 receptor activity of 4-(n-alkyl)-1H-imidazoles and 4-(omega-phenylalkyl)-1H-imidazoles

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https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Synthesis of potent non-imidazole histamine H3-receptor antagonists.

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https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Sensitive radioimmunoassays for histamine and tele-methylhistamine in the brain

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7 January 2021

Synthesis of new potent and selective aromatase inhibitors based on long-chained diarylalkylimidazole and diarylalkyltriazole molecule skeletons

1 reference

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7 January 2021

Pyrazoles as potential histamine H3-receptor antagonists

1 reference

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7 January 2021

Azines and diazines as potential histamine H3-receptor antagonists

1 reference

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7 January 2021

Therapeutic potential of histamine H3 receptor agonists and antagonists.

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https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Design, synthesis, and structure-activity relationships of novel non-imidazole histamine H(3) receptor antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

The Use of Diethyl Azodicarboxylate and Triphenylphosphine in Synthesis and Transformation of Natural Products

1 reference

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7 January 2021

Effects of thioperamide, a histamine H3-receptor antagonist, on a scopolamine-induced learning deficit using an elevated plus-maze test in mice

1 reference

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7 January 2021

Inhibition of histamine versus acetylcholine metabolism as a mechanism of tacrine activity.

1 reference

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7 January 2021

Reduction of organic compounds by lithium aluminum hydride; halides, quinones, miscellaneous nitrogen compounds

1 reference

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7 January 2021

Improvement by FUB 181, a novel histamine H3-receptor antagonist, of learning and memory in the elevated plus-maze test in mice.

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Heteroarylaminoethyl and heteroarylthioethyl imidazoles. Synthesis and H3-receptor affinity

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Development of chiral N-alkylcarbamates as new leads for potent and selective H3-receptor antagonists: synthesis, capillary electrophoresis, and in vitro and oral in vivo activity.

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Novel histamine H3 receptor antagonists: affinities in an H3 receptor binding assay and potencies in two functional H3 receptor models

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

The moderate affinity of clozapine at H3 receptors is not shared by its two major metabolites and by structurally related and unrelated atypical neuroleptics.

1 reference

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7 January 2021

Histaminergic transmission in the mammalian brain

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https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Novel carbamates as potent histamine H3 receptor antagonists with high in vitro and oral in vivo activity

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Development of FUB 181, a selective histamine H3-receptor antagonist of high oral in vivo potency with 4-(omega-(arylalkyloxy)alkyl)-1H-imidazole structure.

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

General construction pattern of histamine H3-receptor antagonists: change of a paradigm

1 reference

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7 January 2021

Novel histamine H(3)-receptor antagonists with carbonyl-substituted 4-(3-(phenoxy)propyl)-1H-imidazole structures like ciproxifan and related compounds

1 reference

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7 January 2021

Cloning and cerebral expression of the guinea pig histamine H3 receptor: evidence for two isoforms

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Homologs of histamine as histamine H3 receptor antagonists: a new potent and selective H3 antagonist, 4(5)-(5-aminopentyl)-1H-imidazole

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Non-imidazole histamine H3 ligands. Part I. Synthesis of 2-(1-piperazinyl)- and 2-(hexahydro-1H-1,4-diazepin-1-yl)benzothiazole derivatives as H3-antagonists with H1 blocking activities

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Non-imidazole histamine H3 ligands, Part 2: New 2-substituted benzothiazoles as histamine H3 antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Some properties of synaptic membranes isolated from the central nervous system

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Effect of thioperamide, a histamine H3 receptor antagonist, on electrically induced convulsions in mice.

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

Clobenpropit (VUF-9153), a new histamine H3 receptor antagonist, inhibits electrically induced convulsions in mice.

1 reference

https://api.crossref.org/works/10.1016%2FS0928-0987%2801%2900106-3

7 January 2021

10.1016/S0928-0987(01)00106-3

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DOI

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25 November 2017

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