Characterization of three non-peptide endothelin receptor ligands using human cloned ETA and ETB receptors (Q42243584)

19 October 2017

Characterization of three non-peptide endothelin receptor ligands using human cloned ETA and ETB receptors (English)

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19 October 2017

Buchan KW

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19 October 2017

Alldus C

2

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19 October 2017

Christodoulou C

3

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19 October 2017

Clark KL

4

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19 October 2017

Dykes CW

5

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19 October 2017

Sumner MJ

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19 October 2017

Wallace DM

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19 October 2017

White DG

8

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19 October 2017

Watts IS

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19 October 2017

language of work or name

English

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publication date

1 August 1994

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British Journal of Pharmacology

19 October 2017

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19 October 2017

112

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19 October 2017

4

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19 October 2017

1251-1257

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A novel ETA-receptor antagonist, FR 139317, inhibits endothelin-induced contractions of guinea-pig pulmonary arteries, but not trachea

19 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Molecular characterization and regulation of the human endothelin receptors

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

The discovery of sulfonamide endothelin antagonists and the development of the orally active ETA antagonist 5-(dimethylamino)-N-(3,4-dimethyl-5-isoxazolyl)-1-naphthalenesulf onamide.

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

In vitro characterization of Ro 46-2005, a novel synthetic non-peptide endothelin antagonist of ETA and ETB receptors

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Endothelin ETA and ETB receptors mediate vascular smooth-muscle contraction

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Quantitative analysis of drug-receptor interactions: I. Determination of kinetic and equilibrium properties

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Endothelin, a novel endothelium-derived peptide. Pharmacological activities, regulation and possible roles in cardiovascular control

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Endothelium-dependent vascular activities of endothelin-like peptides in the isolated superior mesenteric arterial bed of the rat

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Cloning of a cDNA encoding a non-isopeptide-selective subtype of the endothelin receptor

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Cloning and expression of a cDNA encoding an endothelin receptor

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Cloning and characterization of cDNA encoding human a-type endothelin receptor

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Cloning and functional expression of human cDNA for the ETB endothelin receptor

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Kinetic analyses demonstrate that the equilibrium assumption does not apply to [125I]endothelin-1 binding data

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Molecular characterization of endothelin receptors

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Binding of [125I]-endothelin-1 to rat cerebellar homogenates and its interactions with some analogues

26 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Sarafotoxin S6c: An agonist which distinguishes between endothelin receptor subtypes

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

[Ala1,3,11,15]endothelin-1 analogs with ETB agonistic activity.

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Endothelin ETA and ETB receptors mediate vascular smooth muscle contraction

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Contractile actions of endothelin-1 in isolated helical strips from rat pulmonary artery: potentiation of serotonin-induced contraction

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Biological profiles of highly potent novel endothelin antagonists selective for the ETA receptor

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Simultaneous analysis of families of sigmoidal curves: application to bioassay, radioligand assay, and physiological dose-response curves

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Use of the endothelin antagonists BQ-123 and PD 142893 to reveal three endothelin receptors mediating smooth muscle contraction and the release of EDRF.

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910249

Molecular Cloning of Human Endothelin (ET) Receptors ETA and ETB

17 August 2018

1 reference

Crossref

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1994.TB13218.X

Pathophysiological role of endothelin revealed by the first orally active endothelin receptor antagonist

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1994.TB13218.X

Endothelin and structurally related analogs distinguish between endothelin receptor subtypes

21 January 2018

1 reference

12 December 2020

Coupling of two endothelin receptor subtypes to differing signal transduction in transfected Chinese hamster ovary cells

1 reference

12 December 2020

Characterization of rat lung endothelin receptor subtypes which are coupled to phosphoinositide hydrolysis

1 reference

12 December 2020

The endothelin family of peptides: local hormones with diverse roles in health and disease?

1 reference

12 December 2020

Human placental membranes contain predominantly ETB receptors

1 reference

12 December 2020

The activity of peptides of the endothelin family in various mammalian smooth muscle preparations

1 reference

12 December 2020

10.1111/J.1476-5381.1994.TB13218.X

Identifiers

DOI

1 reference

19 October 2017

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19 October 2017

PubMed publication ID

7952888

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