Compared pharmacology of human histamine H3 and H4 receptors: structure-activity relationships of histamine derivatives (Q41888634)

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15 January 2020

title

Compared pharmacology of human histamine H3 and H4 receptors: structure-activity relationships of histamine derivatives (English)

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15 January 2020

3

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15 January 2020

author name string

Florence Gbahou

1

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15 January 2020

Ludwig Vincent

2

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15 January 2020

Joel Tardivel-Lacombe

4

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15 January 2020

Claude Chabret

5

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15 January 2020

Jean-Michel Arrang

6

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15 January 2020

language of work or name

English

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publication date

1 April 2006

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British Journal of Pharmacology

15 January 2020

published in

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15 January 2020

volume

147

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15 January 2020

page(s)

744-754

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15 January 2020

issue

7

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The histamine H4 receptor as a new therapeutic target for inflammation

15 January 2020

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Histamine h(4) and h(2) receptors control histamine-induced interleukin-16 release from human CD8(+) T cells

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A detailed mapping of the histamine H(3) receptor and its gene transcripts in rat brain

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Molecular modeling and site-specific mutagenesis of the histamine-binding site of the histamine H4 receptor.

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cDNA cloning and characterization of porcine histamine H4 receptor

5 June 2018

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Histamine H3-receptor-mediated [35S]GTP gamma[S] binding: evidence for constitutive activity of the recombinant and native rat and human H3 receptors.

5 June 2018

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Comparison of human, mouse, rat, and guinea pig histamine H4 receptors reveals substantial pharmacological species variation

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Genomic organization and characterization of splice variants of the human histamine H3 receptor

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5 June 2018

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Cloning and pharmacological characterization of a fourth histamine receptor (H(4)) expressed in bone marrow

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Genomics meets histamine receptors: new subtypes, new receptors.

5 June 2018

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The rat H3 receptor: gene organization and multiple isoforms.

5 June 2018

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High constitutive activity of native H3 receptors regulates histamine neurons in brain.

5 June 2018

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Molecular cloning and characterization of a new human histamine receptor, HH4R

5 June 2018

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Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain

5 June 2018

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Molecular cloning and characterization of a novel type of histamine receptor preferentially expressed in leukocytes

5 June 2018

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5 June 2018

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Cloning and functional expression of the human histamine H3 receptor

5 June 2018

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5 June 2018

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Differential effect of sodium ions and guanine nucleotides on the binding of thioperamide and clobenpropit to histamine H3-receptors in rat cerebral cortical membranes

5 June 2018

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Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

5 June 2018

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Definition and antagonism of histamine H 2 -receptors

5 June 2018

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

5 June 2018

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Highly potent and selective ligands for histamine H3-receptors

5 June 2018

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H3-receptors control histamine release in human brain

5 June 2018

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Stereoselectivity of the histamine H3-presynaptic autoreceptor

5 June 2018

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Reversible and irreversible labeling and autoradiographic localization of the cerebral histamine H2 receptor using [125I]iodinated probes

5 June 2018

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5 June 2018

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Histamine H3 receptor binding sites in rat brain membranes: modulations by guanine nucleotides and divalent cations

5 June 2018

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Characterisation of the binding of the histamine H3 receptor agonist [3H] (R)-alpha methyl histamine to homogenates of rat and guinea-pig cortex.

5 June 2018

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Synthesis, absolute configuration, stereoselectivity, and receptor selectivity of (.alpha.R,.beta.S)-.alpha.,.beta.-dimethylhistamine. A novel highly potent histamine H3 receptor agonist

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Specific binding of 3H-mepyramine to histamine H1 receptors in intestinal smooth muscle

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Critical Role of Histamine H4Receptor in Leukotriene B4Production and Mast Cell-Dependent Neutrophil Recruitment Induced by Zymosan in Vivo

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Generation and characterization of highly constitutive active histamine H3 receptors

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The role of transmembrane helix 5 in agonist binding to the human H3 receptor

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Constitutive activity of histamine h(3) receptors stably expressed in SK-N-MC cells: display of agonism and inverse agonism by H(3) antagonists

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Identification of rat H3 receptor isoforms with different brain expression and signaling properties.

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The profiles of human and primate [3H]Nalpha-methylhistamine binding differ from that of rodents.

18 August 2018

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Pharmacological estimation of drug-receptor dissociation constants. Statistical evaluation. I. Agonists

18 August 2018

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[125I]iodoproxyfan, a new antagonist to label and visualize cerebral histamine H3 receptors

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PubMed

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inferred from PubMed ID database lookup

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Identifiers

DOI

10.1038/SJ.BJP.0706666

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:16432504%20AND%20SRC:MED&resulttype=core&format=json

15 January 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:16432504%20AND%20SRC:MED&resulttype=core&format=json

15 January 2020

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