Pharmacological properties of recombinant "diazepam-insensitive" GABAA receptors (Q41243374)

28 September 2017

Pharmacological properties of recombinant "diazepam-insensitive" GABAA receptors (English)

1 reference

28 September 2017

0 references

Gunnersen D

1

1 reference

28 September 2017

Kaufman CM

series ordinal

2

1 reference

28 September 2017

Skolnick P

series ordinal

3

1 reference

28 September 2017

1 January 1996

1 reference

28 September 2017

8

1 reference

based on heuristic

inferred from page(s)

published in

Neuropharmacology

1 reference

28 September 2017

35

1 reference

28 September 2017

9-10

1 reference

28 September 2017

1307-1314

1 reference

Beta-carbolines: synthesis and neurochemical and pharmacological actions on brain benzodiazepine receptors.

28 September 2017

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Triazolam is more efficacious than diazepam in a broad spectrum of recombinant GABAA receptors.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Synthesis and evaluation of imidazo[1,5-a][1,4]benzodiazepine esters with high affinities and selectivities at "diazepam-insensitive" benzodiazepine receptors.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Contribution of "diazepam-insensitive" GABAA receptors to the alcohol antagonist properties of Ro 15-4513 and related imidazobenzodiazepines.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Characterization of diazepam-insensitive [3H]Ro 15-4513 binding in rodent brain and cultured cerebellar neuronal cells.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Novel GABAA receptor alpha subunit is expressed only in cerebellar granule cells.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

The subunit composition of a GABAA/benzodiazepine receptor from rat cerebellum.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Current potentiation by diazepam but not GABA sensitivity is determined by a single histidine residue.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Natural mutation of GABAA receptor alpha 6 subunit alters benzodiazepine affinity but not allosteric GABA effects

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Substrate specificity of diazepan-insensitive cerebellar [3H] Ro 15-4513 binding sites

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Benzodiazepine-induced motor impairment linked to point mutation in cerebellar GABAA receptor.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Antagonism of the intoxicating effects of ethanol by the potent benzodiazepine receptor ligand Ro 19-4603

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Cerebellar GABAA receptor selective for a behavioural alcohol antagonist

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Diazepam-insensitive [3H]Ro 15-4513 binding in intact cultured cerebellar granule cells.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Importance of a novel GABAA receptor subunit for benzodiazepine pharmacology

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Photoaffinity labeling of benzodiazepine receptor proteins with the partial inverse agonist [3H]Ro 15-4513: a biochemical and autoradiographic study.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

A selective imidazobenzodiazepine antagonist of ethanol in the rat.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Ethanol stimulates gamma-aminobutyric acid receptor-mediated chloride transport in rat brain synaptoneurosomes

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Ro15-4513 differentially affects ethanol-induced hypnosis and hypothermia.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Diazepam sensitivity of the binding of an imidazobenzodiazepine, [3H]Ro 15-4513, in cerebellar membranes from two rat lines developed for high and low alcohol sensitivity

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Functional properties of recombinant rat GABAA receptors depend upon subunit composition

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Four amino acid exchanges convert a diazepam-insensitive, inverse agonist-preferring GABAA receptor into a diazepam-preferring GABAA receptor

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Cloning, pharmacological characteristics and expression pattern of the rat GABAA receptor alpha 4 subunit

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

The distribution of 13 GABAA receptor subunit mRNAs in the rat brain. I. Telencephalon, diencephalon, mesencephalon

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

High affinity ligands for ‘diazepam-insensitive’ benzodiazepine receptors

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Ro 15-4513 binding to GABAA receptors: subunit composition determines ligand efficacy

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Labelling of diazepam-sensitive and -insensitive benzodiazepine receptors with [3H]tert-butyl-8-chloro-5,6-dihydro-5-methyl-6-oxo-4H-imidazo [1,5-a][1,4]benzodiazepine 3-carboxylate (ZG-63).

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Synthetic and computer-assisted analysis of the structural requirements for selective, high-affinity ligand binding to diazepam-insensitive benzodiazepine receptors.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Cloning and characterization of the human GABAA receptor alpha 4 subunit: identification of a unique diazepam-insensitive binding site

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Sequence and expression of a novel GABAA receptor alpha subunit.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

Synthesis of novel imidazobenzodiazepines as probes of the pharmacophore for "diazepam-insensitive" GABAA receptors

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2896%2900054-8

10.1016/S0028-3908(96)00054-8

7 January 2021

Identifiers

DOI

1 reference

release_tg6xj6kak5ah3cl6cdspxfejl4

28 September 2017

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/tg6xj6kak5ah3cl6cdspxfejl4

mapped directly with Wikidata item

24 November 2022

based on heuristic

1 reference