5-HT1A receptor agonists: recent developments and controversial issues (Q40933736)

25 September 2017

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title

5-HT1A receptor agonists: recent developments and controversial issues (English)

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25 September 2017

J De Vry

1

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25 September 2017

1 September 1995

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25 September 2017

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25 September 2017

121

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25 September 2017

1-26

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25 September 2017

1

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https://scigraph.springernature.com/pub.10.1007/bf02245588

25 September 2017

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cites work

Effect of chronic treatment with 5-HT1 agonist (8-OH-DPAT and RU 24969) and antagonist (isapirone) drugs on the behavioural responses of mice to 5-HT1 and 5-HT2 agonists

1 reference

https://api.crossref.org/works/10.1007%2FBF02245588

The effect of dinoprost on transport of water and imipramine through rat small intestinal membranes

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FBF02245588

Differential effects of centrally-active antihypertensives on 5-HT1A receptors in rat dorso-lateral septum, rat hippocampus and guinea-pig hippocampus

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FBF02245588

Mediation of the antidepressant-like effect of 8-OH-DPAT in mice by postsynaptic 5-HT1A receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FBF02245588

Adaptive changes in 5-HT1A receptor-mediated hippocampal inhibition in the alert rat produced by repeated 8-OH-DPAT treatment.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FBF02245588

Characterization of 8-OH-DPAT-induced hypothermia in mice as a 5-HT1A autoreceptor response and its evaluation as a model to selectively identify antidepressants

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FBF02245588

Reversal of neuroleptic-induced catalepsy by novel aryl-piperazine anxiolytic drugs

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FBF02245588

Corticosterone suppresses the expression of 5-HT1A receptor mRNA in rat dentate gyrus.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FBF02245588

Actions of 5-HT1 ligands on excitatory synaptic transmission in the hippocampus of alert rats

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FBF02245588

Different effects of intracerebral and systemic administration of buspirone in the forced swimming test: involvement of a metabolite.

21 January 2018

1 reference

12 December 2020

Comparison of 5-hydroxytryptamine1A-mediated hyperpolarization in CA1 and CA3 hippocampal pyramidal cells

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12 December 2020

Effect of 5-HT1A receptor agonists in two models of anxiety after dorsal raphe injection

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12 December 2020

Heterogeneity of cortical and hippocampal 5-HT1A receptors: a reappraisal of homogenate binding with 8-[3H]hydroxydipropylaminotetralin.

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12 December 2020

Ipsapirone and 8-OH-DPAT reduce ethanol preference in rats: involvement of presynaptic 5-HT1A receptors.

1 reference

12 December 2020

Stimulation of hippocampal 5-HT1A receptors causes amnesia and anxiolytic-like but not antidepressant-like effects in the rat.

1 reference

12 December 2020

Molecular biology of serotonin (5-HT) receptors

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12 December 2020

5-HT receptors as targets for the development of novel anxiolytic drugs: models, mechanisms and future directions

1 reference

12 December 2020

Involvement of the dorsal hippocampus in mediation of the antianxiety action of tandospirone, a 5-hydroxytryptamine1A agonistic anxiolytic

1 reference

12 December 2020

Effects of 5-HT-1A receptor agonists on ethanol preference in the rat

1 reference

12 December 2020

Lack of apparent receptor reserve at postsynaptic 5-hydroxytryptamine1A receptors negatively coupled to adenylyl cyclase activity in rat hippocampal membranes

1 reference

12 December 2020

Differential properties of pre- and postsynaptic 5-hydroxytryptamine1A receptors in the dorsal raphe and hippocampus: I. Effect of spiperone.

1 reference

12 December 2020

A study of the mechanism of Ca2+ current inhibition produced by serotonin in rat dorsal raphe neurons

1 reference

12 December 2020

Serotonin 5-HT1A receptor-mediated hypothermia in mice: absence of spare receptors and rapid induction of tolerance

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12 December 2020

International Union of Pharmacology classification of receptors for 5-hydroxytryptamine (Serotonin)

1 reference

12 December 2020

Long-Term Antidepressant Treatment Decreases Spiroperidol-Labeled Serotonin Receptor Binding

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12 December 2020

The relation of central 5-HT1A and 5-HT2 receptors: Low dose agonist-induced selective tolerance in the rat

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12 December 2020

Anxiolytic effects of the 5-HT1A receptor agonist ipsapirone in the rat: neurobiological correlates.

1 reference

12 December 2020

Effect of metergoline, fenfluramine, and 8-OHDPAT on catalepsy induced by haloperidol or morphine

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12 December 2020

Differential properties of pre- and postsynaptic 5-hydroxytryptamine1A receptors in the dorsal raphe and hippocampus: II. Effect of pertussis and cholera toxins.

1 reference

12 December 2020

Shock-induced ultrasonic vocalization in young adult rats: a model for testing putative anti-anxiety drugs

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12 December 2020

Antidepressant-like behavioral effects of serotonin receptor agonists

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12 December 2020

The long-term effects of 8-hydroxy-2-(di-n-propyl-amino)tetralin (8-OH-DPAT) on copulatory and exploratory behaviour in male rats

1 reference

12 December 2020

Alterations of central serotoninergic and dopaminergic neurotransmission in rats chronically treated with ipsapirone: biochemical and electrophysiological studies

1 reference

12 December 2020

Alterations of central serotonin and dopamine turnover in rats treated with ipsapirone and other 5-hydroxytryptamine1A agonists with potential anxiolytic properties

1 reference

12 December 2020

Antipsychotic-like profile of combined treatment with raclopride and 8-OH-DPAT in the rat: enhancement of antipsychotic-like effects without catalepsy

1 reference

12 December 2020

5-HT1A-sensitive adenylyl cyclase of rodent hippocampal neurons: effects of antidepressant treatments and chronic stimulation with agonists

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12 December 2020

5-HT1A receptor influences on rodent social and agonistic behavior: a review and empirical study

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12 December 2020

Silent 5-HT1A receptor antagonists: utility as research tools and therapeutic agents.

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12 December 2020

Ipsapirone depresses neuronal activity in the dorsal raphe nucleus and the hippocampal formation.

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12 December 2020

Antidepressant-like effects of buspirone mediated by the 5-HT1A post-synaptic receptors in the learned helplessness paradigm.

1 reference

12 December 2020

Alcohol drinking in rats treated with 5,7-dihydroxytryptamine: effect of 8-OH-DPAT and tropisetron (ICS 205-930).

1 reference

12 December 2020

Involvement of the serotonergic system in ethanol intake in the rat.

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12 December 2020

5-HT1A receptor ligands in animal models of anxiety, impulsivity and depression: multiple mechanisms of action?

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12 December 2020

Isapirone is a partial agonist at 5-hydroxytryptamine 1A (5-HT1A) receptors in the rat hippocampus: electrophysiological evidence.

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12 December 2020

Effect of chronic treatment with 8-OH-DPAT in the forced swimming test requires the integrity of presynaptic serotonergic mechanisms.

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12 December 2020

A comparison of the effects of diazepam versus several typical and atypical anti-depressant drugs in an animal model of anxiety

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12 December 2020

(-)Tertatolol is a potent antagonist at pre- and postsynaptic serotonin 5-HT1A receptors in the rat brain.

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12 December 2020

Effect of acute and chronic treatment of rats with the putative anxiolytic drug ipsapirone on the turnover of monoamine transmitters in various brain regions. A comparison with the 5-HT1A agonist 8-OH-DPAT.

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12 December 2020

Increase of extracellular dopamine in the prefrontal cortex: a trait of drugs with antidepressant potential?

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12 December 2020

Neuroanatomical basis for the antidepressant-like effects of the 5-HT(1A) receptor agonists 8-OH-DPAT and ipsapirone in the rat forced swimming test

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12 December 2020

Effect of chronic treatments with tandospirone and imipramine on serotonin-mediated behavioral responses and monoamine receptors.

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12 December 2020

Convergence and divergence of neurotransmitter action in human cerebral cortex

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12 December 2020

Comparative effects of chronic 8-OH-DPAT, gepirone and ipsapirone treatment on the sensitivity of somatodendritic 5-HT1A autoreceptors.

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12 December 2020

Tandospirone and its metabolite, 1-(2-pyrimidinyl)-piperazine--I. Effects of acute and long-term administration of tandospirone on serotonin neurotransmission.

1 reference

12 December 2020

Effect of chronic treatment on the cardiovascular and behavioral responses of 8-OH-DPAT in conscious normotensive rats

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12 December 2020

The effects of a 5-HT1 receptor ligand isapirone (TVX Q 7821) on 5-HT synthesis and the behavioural effects of 5-HT agonists in mice and rats.

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12 December 2020

8-OH-DPAT suppresses vomiting in the cat elicited by motion, cisplatin or xylazine

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12 December 2020

Increased population spike amplitude in the dentate gyrus following systemic administration of 5-hydroxytryptophan or 8-hydroxy-2-(di-n-propylamino)tetralin

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12 December 2020

5-HT1A receptor-mediated inhibition in the hippocampus of the alert rat — effects of repeated gepirone treatment

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12 December 2020

Chronic treatment with an anxiolytic dose of the 5-HT1A agonist ipsapirone does not alter ipsapirone acute neuroendocrine effects.

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12 December 2020

Effects of the 5-HT receptor agonist, 8-OH-DPAT, on ethanol preference in the rat.

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12 December 2020

Desensitization of 5-HT1A autoreceptors by chronic administration of 8-OH-DPAT

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12 December 2020

5-HT1A receptors activate a potassium conductance in rat ventromedial hypothalamic neurones

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12 December 2020

A single dose of 8-OH-DPAT reduces raphe binding of [3H]8-OH-DPAT and increases the effect of raphe stimulation on 5-HT metabolism

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12 December 2020

Studies on the neuronal circuits involved in the discriminative stimulus effects of 5-hydroxytryptamine1A receptor agonists in the rat.

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12 December 2020

Voluntary intake of alcohol is attenuated by ipsapirone in mice and role of 5-HT1A receptor

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12 December 2020

Effect of drugs influencing 5-HT function on ethanol drinking and feeding behaviour in rats: studies using a drinkometer system.

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12 December 2020

The inhibitory effect of 8-OH-DPAT on the firing activity of dorsal raphe serotoninergic neurons in rats is attenuated by lesion of the frontal cortex.

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12 December 2020

Sex difference for tolerance of 5-HT1A receptor-mediated temperature and corticosterone responses in mice.

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12 December 2020

Aggression, anxiety and vocalizations in animals: GABAA and 5-HT anxiolytics.

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12 December 2020

Differential modulation of three separate K-conductances in hippocampal CA1 neurons by serotonin

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12 December 2020

Single administration of 5-HT1A agonists decreases 5-HT1A presynaptic, but not postsynaptic receptor-mediated responses: relationship to antidepressant-like action

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12 December 2020

Autoradiographic quantification of serotonin1A receptors in rat brain following antidepressant drug treatment

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12 December 2020

Serotonergic innervation of the hippocampus and nucleus accumbens septi and the anxiolytic-like action of midazolam and 5-HT1A receptor agonists.

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12 December 2020

5-HT1A receptors in the median raphe nucleus and dorsal hippocampus may mediate anxiolytic and anxiogenic behaviours respectively.

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12 December 2020

The role of postsynaptic 5-HT1A receptors in the anticonflict effect of ipsapirone.

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12 December 2020

The non-competitive NMDA receptor antagonist (+)MK-801 counteracts the long-lasting attenuation of the hypothermic response induced by acute doses of 8-OH-DPAT in the rat

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12 December 2020

Reduction in cortical 5HT2 receptor sensitivity after continuous gepirone treatment.

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12 December 2020

Reduction of in vivo striatal 5-hydroxytryptamine release by 8-OH-DPAT after inactivation of Gi/G(o) proteins in dorsal raphe nucleus

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12 December 2020

Responses of hippocampal pyramidal cells to putative serotonin 5-HT1A and 5-HT1B agonists: a comparative study with dorsal raphe neurons

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12 December 2020

Influence of the 5-HT1A receptor agonist ipsapirone on voluntary alcohol intake in rats.

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12 December 2020

Neuroprotective properties of 5-HT1A receptor agonists in rodent models of focal and global cerebral ischemia

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12 December 2020

Modification of 5-HT neuron properties by sustained administration of the 5-HT1A agonist gepirone: electrophysiological studies in the rat brain.

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12 December 2020

Pharmacology of 5-hydroxytryptamine-1A receptors which inhibit cAMP production in hippocampal and cortical neurons in primary culture.

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12 December 2020

Effect of acute and repeated administration of 5-HT1A receptor agonists on 5-HT release in rat brain in vivo

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12 December 2020

Repeated treatment with the 5-HT1A receptor agonist, ipsapirone, does not affect 8-OH-DPAT- and stress-induced increases in plasma adrenaline levels in the rat

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12 December 2020

Potential antidepressant properties of 8-hydroxy-2-(di-n-propylamino)tetralin, a selective serotonin1A receptor agonist

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12 December 2020

The effects of long-term treatment with 8-OH-DPAT on the lordosis response and hypothermia in female rate

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12 December 2020

Different effects on the responses of functional pre- and postsynaptic 5-HT1A receptors by repeated treatment of rats with the 5-HT1A receptor agonist 8-OH-DPAT

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12 December 2020

Behavioural and biochemical consequences following activation of 5HT1-like and GABA receptors in the dorsal raphé nucleus of the rat.

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12 December 2020

Median and dorsal raphe injections of the 5-HT1A agonist, 8-OH-DPAT, and the GABAA agonist, muscimol, increase voluntary ethanol intake in Wistar rats.

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12 December 2020

Effects of blockade of 5-HT2 receptors and activation of 5-HT1A receptors on the exploratory activity of rats in the elevated plus-maze.

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12 December 2020

Potential anxiolytic properties of 8-hydroxy-2-(di-n-propylamino)tetralin, a selective serotonin 1A receptor agonist.

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12 December 2020

Alteration of 5-HT1A receptor binding sites following chronic treatment with ipsapirone measured by quantitative autoradiography.

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12 December 2020

Contrasting behavioural effects of 8-OH DPAT in the dorsal raphé nucleus and ventral hippocampus.

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12 December 2020

Biochemical evidence for the regulation of central noradrenergic activity by 5-HT1A and 5-HT2 receptors: microdialysis studies in the awake and anaesthetized rat.

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12 December 2020

Subchronic treatment with anxiolytic doses of the 5-HT1A receptor agonist ipsapirone does not affect 5-HT2 receptor sensitivity in the rat

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12 December 2020

Long lasting attenuation of 8-OH-DPAT-induced corticosterone secretion after a single injection of a 5-HT1A receptor agonist

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12 December 2020

Evidence that the amygdala is involved in benzodiazepine and serotonergic effects on punished responding but not on discrimination.

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12 December 2020

Regulation of 5-hydroxytryptamine1A receptor function in rat hippocampus by short- and long-term administration of 5-hydroxytryptamine1A agonist and antidepressants

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12 December 2020

Neurochemical changes in pigeon cerebrospinal fluid during chronic administration of buspirone or 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT).

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12 December 2020

Agonist/antagonist interactions with cloned human 5-HT1A receptors: variations in intrinsic activity studied in transfected HeLa cells

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12 December 2020

Neuronal circuits involved in the anxiolytic effects of the 5-HT1A receptor agonists 8-OH-DPAT ipsapirone and buspirone in the rat.

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12 December 2020

Are postsynaptic 5-HT1A receptors involved in the anxiolytic effects of 5-HT1A receptor agonists and in their inhibitory effects on the firing of serotonergic neurons in the rat?

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12 December 2020

Antiemetic effects of 5-HT1A agonists in the pigeon.

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12 December 2020

Receptor reserve for 5-hydroxytryptamine1A-mediated inhibition of serotonin synthesis: possible relationship to anxiolytic properties of 5-hydroxytryptamine1A agonists.

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12 December 2020

5HT drugs in animal models of anxiety

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12 December 2020

Neurophysiological effects of buspirone and isapirone in the hippocampus: comparison with 5-hydroxytryptamine.

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12 December 2020

Low doses of the 5-HT1A agonist 8-hydroxy-2-(di-n-propylamino)-tetralin (8-OH DPAT) increase ethanol intake

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12 December 2020

Serotonin, dopamine and GABA involvement in alcohol drinking of selectively bred rats

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12 December 2020

The effects of acute administration of gepirone in rats trained on conflict schedules having different degrees of predictability.

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12 December 2020

8-Hydroxy-2-(di-n-propylamino)tetralin, a selective serotonin1A receptor agonist, reduces the immobility of rats in the forced swimming test by acting on the nucleus raphe dorsalis.

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12 December 2020

5-Hydroxytryptamine2 and 5-hydroxytryptamine1A receptors mediate opposing responses on membrane excitability in rat association cortex

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12 December 2020

Unique modulation of central 5-HT2 receptor binding sites and 5-HT2 receptor-mediated behavior by continuous gepirone treatment

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12 December 2020

Identifiers

DOI

10.1007/BF02245588

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PubMed ID

8539333

Dimensions Publication ID

25 September 2017

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PubMed ID

8539333