Conformational States of HIV-1 Reverse Transcriptase for Nucleotide Incorporation vs Pyrophosphorolysis-Binding of Foscarnet. (Q40748250)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27192549%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

title

Conformational States of HIV-1 Reverse Transcriptase for Nucleotide Incorporation vs Pyrophosphorolysis-Binding of Foscarnet (English)

1 reference

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2 April 2020

4

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2 April 2020

Kalyan Das

1

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2 April 2020

author name string

Jan Balzarini

2

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2 April 2020

Matthew T Miller

3

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2 April 2020

Jeffrey J DeStefano

5

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2 April 2020

Eddy Arnold

6

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2 April 2020

publication date

6 June 2016

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2 April 2020

1 reference

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2 April 2020

volume

11

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2 April 2020

page(s)

2158-2164

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2 April 2020

issue

8

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Exploring the role of the α-carboxyphosphonate moiety in the HIV-RT activity of α-carboxy nucleoside phosphonates

2 April 2020

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The pyrophosphate analogue foscarnet traps the pre-translocational state of HIV-1 reverse transcriptase in a Brownian ratchet model of polymerase translocation

24 September 2017

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Indolopyridones inhibit human immunodeficiency virus reverse transcriptase with a novel mechanism of action

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24 September 2017

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24 September 2017

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24 September 2017

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24 September 2017

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24 September 2017

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24 September 2017

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24 September 2017

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24 September 2017

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24 September 2017

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24 September 2017

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24 September 2017

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24 September 2017

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15 June 2018

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15 June 2018

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15 June 2018

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17 June 2018

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Mechanism by which phosphonoformic acid resistance mutations restore 3'-azido-3'-deoxythymidine (AZT) sensitivity to AZT-resistant HIV-1 reverse transcriptase.

19 August 2018

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19 August 2018

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Roles of Conformational and Positional Adaptability in Structure-Based Design of TMC125-R165335 (Etravirine) and Related Non-nucleoside Reverse Transcriptase Inhibitors That Are Highly Potent and Effective against Wild-Type and Drug-Resistant HIV-1 V

2 December 2018

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HIV resistance to zidovudine: the role of pyrophosphorolysis

2 December 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/27192549

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Site-directed mutagenesis of arginine 72 of HIV-1 reverse transcriptase. Catalytic role and inhibitor sensitivity

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/27192549

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/ACSCHEMBIO.6B00187

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27192549%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27192549%20AND%20SRC:MED&resulttype=core&format=json

2 April 2020

1 reference