Asymmetric functioning of dimeric metabotropic glutamate receptors disclosed by positive allosteric modulators. (Q40428691)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15863499%20AND%20SRC:MED&resulttype=core&format=json

11 January 2020

title

Asymmetric functioning of dimeric metabotropic glutamate receptors disclosed by positive allosteric modulators (English)

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11 January 2020

1

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11 January 2020

Julie Kniazeff

2

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11 January 2020

Damien Maurel

5

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11 January 2020

Jaroslav Blahoš

7

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11 January 2020

Jean-Philippe Pin

9

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11 January 2020

author name string

Veronika Hlavackova

3

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11 January 2020

Fanny Malhaire

4

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11 January 2020

Francine Acher

6

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11 January 2020

Laurent Prézeau

8

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11 January 2020

language of work or name

English

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publication date

29 April 2005

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Journal of Biological Chemistry

11 January 2020

published in

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11 January 2020

volume

280

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11 January 2020

issue

26

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11 January 2020

page(s)

24380-24385

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Evidence for a single heptahelical domain being turned on upon activation of a dimeric GPCR

11 January 2020

cites work

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Heptahelical domain of metabotropic glutamate receptor 5 behaves like rhodopsin-like receptors.

22 September 2017

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The calcimimetic cinacalcet normalizes serum calcium in subjects with primary hyperparathyroidism

22 September 2017

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22 September 2017

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Pharmacological characterization and identification of amino acids involved in the positive modulation of metabotropic glutamate receptor subtype 2.

22 September 2017

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A family of highly selective allosteric modulators of the metabotropic glutamate receptor subtype 5.

22 September 2017

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Structure-based analysis of GPCR function: evidence for a novel pentameric assembly between the dimeric leukotriene B4 receptor BLT1 and the G-protein

22 September 2017

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Evolution, structure, and activation mechanism of family 3/C G-protein-coupled receptors

22 September 2017

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Organization of the G protein-coupled receptors rhodopsin and opsin in native membranes

22 September 2017

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Closure of the Venus flytrap module of mGlu8 receptor and the activation process: Insights from mutations converting antagonists into agonists

22 September 2017

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22 September 2017

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Structural views of the ligand-binding cores of a metabotropic glutamate receptor complexed with an antagonist and both glutamate and Gd3+.

22 September 2017

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22 September 2017

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22 September 2017

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22 September 2017

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Structural basis of glutamate recognition by a dimeric metabotropic glutamate receptor

22 September 2017

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22 September 2017

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22 September 2017

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25 September 2017

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17 June 2018

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The second intracellular loop of metabotropic glutamate receptors recognizes C termini of G-protein alpha-subunits.

20 August 2018

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20 August 2018

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20 August 2018

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Metabotropic glutamate receptor 5 is a disulfide-linked dimer

20 August 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/15863499

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1074/JBC.M502642200

1 reference

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11 January 2020

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11 January 2020

1 reference