Novel 1,2-dihydroquinazolin-2-ones: Design, synthesis, and biological evaluation against Trypanosoma brucei (Q38669388)

http://europepmc.org/abstract/PMC/6214665

30 June 2019

title

Novel 1,2-dihydroquinazolin-2-ones: Design, synthesis, and biological evaluation against Trypanosoma brucei (English)

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http://europepmc.org/abstract/PMC/6214665

30 June 2019

main subject

Trypanosoma brucei

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author

Dolores Gonzalez-Pacanowska

17

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5 June 2020

Rosario Díaz González

4

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5 June 2020

Francisco Gamarro

16

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Miguel Navarro

18

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5 June 2020

5

Guiomar Pérez-Moreno

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5 June 2020

Gloria Ceballos-Pérez

6

object named as

Gloria Ceballos-Pérez

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7

Veronica Gomez-Pérez

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author name string

ThanhTruc Pham

1

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Madeline Walden

2

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Christopher Butler

3

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Raquel García-Hernández

8

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Henry Zecca

9

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Emma Krakoff

10

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Brian Kopec

11

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Ogar Ichire

12

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Caden Mackenzie

13

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Marika Pitot

14

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Luis Miguel Ruiz

15

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Amy B Dounay

19

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5 June 2020

language of work or name

English

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publication date

11 July 2017

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http://europepmc.org/abstract/PMC/6214665

30 June 2019

published in

Bioorganic & Medicinal Chemistry Letters

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volume

27

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5 June 2020

page(s)

3629-3635

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issue

16

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PAINS in the assay: chemical mechanisms of assay interference and promiscuous enzymatic inhibition observed during a sulfhydryl-scavenging HTS.

5 June 2020

cites work

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Identification and characterization of hundreds of potent and selective inhibitors of Trypanosoma brucei growth from a kinase-targeted library screening campaign

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Safety and efficacy of the 10-day melarsoprol schedule for the treatment of second stage Rhodesiense sleeping sickness

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12 December 2020

10.1016/J.BMCL.2017.07.032

Identifiers

DOI

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5 June 2020

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