Measuring the tyrosine kinase activity: a review of biochemical and cellular assay technologies (Q38088804)

28 August 2017

title

Measuring the tyrosine kinase activity: a review of biochemical and cellular assay technologies (English)

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28 August 2017

Yong Jia

1

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28 August 2017

Xiang-Ju Gu

series ordinal

2

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28 August 2017

Achim Brinker

series ordinal

3

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28 August 2017

Markus Warmuth

series ordinal

4

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28 August 2017

language of work or name

English

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publication date

1 August 2008

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Expert Opinion on Drug Discovery

28 August 2017

published in

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28 August 2017

volume

3

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28 August 2017

issue

8

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28 August 2017

page(s)

959-978

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The protein kinase complement of the human genome

28 August 2017

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Kinases as therapeutic targets for heart failure

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Detection of protein tyrosine kinase activity using a high-capacity streptavidin-coated membrane and optimized biotinylated peptide substrates

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Identification of inhibitors of the kinase activity of oncogenic V600E BRAF in an enzyme cascade high-throughput screen

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A Widely Applicable, High-Throughput TR-FRET Assay for the Measurement of Kinase Autophosphorylation: VEGFR-2 as a Prototype

21 January 2018

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Assay concordance between SPA and TR-FRET in high-throughput screening

21 January 2018

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Fluorescence polarization competition immunoassay for tyrosine kinases

21 January 2018

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Readout technologies for highly miniaturized kinase assays applicable to high-throughput screening in a 1536-well format.

21 January 2018

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Data Concordance from a Comparison between Filter Binding and Fluorescence Polarization Assay Formats for Identification of ROCK-II Inhibitors

21 January 2018

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An evaluation of fluorescence polarization and lifetime discriminated polarization for high throughput screening of serine/threonine kinases

21 January 2018

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Detection of phosphopeptides by fluorescence polarization in the presence of cationic polyamino acids: application to kinase assays

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Fluorescence polarization and anisotropy in high throughput screening: perspectives and primer

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Miniaturization and validation of a high-throughput serine kinase assay using the AlphaScreen platform

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Further comparison of primary hit identification by different assay technologies and effects of assay measurement variability

21 January 2018

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Development of a fluorescence polarization AKT serine/threonine kinase assay using an immobilized metal ion affinity-based technology

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High-throughput screening with immobilized metal ion affinity-based fluorescence polarization detection, a homogeneous assay for protein kinases

21 January 2018

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A homogeneous fluorescence polarization assay adaptable for a range of protein serine/threonine and tyrosine kinases

21 January 2018

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Using IMAP technology to identify kinase inhibitors: comparison with a substrate depletion approach and analysis of the nature of false positives

21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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A generic, homogenous method for measuring kinase and inhibitor activity via adenosine 5'-diphosphate accumulation

21 January 2018

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Application of meso scale technology for the measurement of phosphoproteins in human tumor xenografts

21 January 2018

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Determination of ligand binding affinities for endogenous seven-transmembrane receptors using fluorometric microvolume assay technology

21 January 2018

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High-throughput cellular assays for regulated posttranslational modifications

21 January 2018

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Cellular Ser/Thr-kinase assays using generic peptide substrates

21 January 2018

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An efficient rapid system for profiling the cellular activities of molecular libraries.

21 January 2018

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Cell-based high-content screening of small-molecule libraries

21 January 2018

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Image-based chemical screening

21 January 2018

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A miniaturized cell-based fluorescence resonance energy transfer assay for insulin-receptor activation.

21 January 2018

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Genetically encoded reporters of protein kinase A activity reveal impact of substrate tethering

21 January 2018

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Genetically encoded fluorescent reporters of protein tyrosine kinase activities in living cells

21 January 2018

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A genetically encoded fluorescent reporter reveals oscillatory phosphorylation by protein kinase C

21 January 2018

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Molecular imaging of Akt kinase activity

21 January 2018

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Transformation of an interleukin 3-dependent hematopoietic cell line by the chronic myelogenous leukemia-specific P210bcr/abl protein

21 January 2018

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Miniaturized, ultra-high throughput screening of tyrosine kinases using homogeneous, competitive fluorescence immunoassays

21 January 2018

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Two simple and generic antibody-independent kinase assays: comparison of a bioluminescent and a microfluidic assay format

21 January 2018

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21 January 2018

Identifiers

DOI

10.1517/17460441.3.8.959

1 reference

release_7glauda2orgulgju54s5jygdm4

28 August 2017

Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/7glauda2orgulgju54s5jygdm4

mapped directly with Wikidata item

24 November 2022

based on heuristic

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