A cannabinoid receptor 1 mutation proximal to the DRY motif results in constitutive activity and reveals intramolecular interactions involved in receptor activation (Q37323369)

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scientific article published on 31 July 2006

Language	Label	Description	Also known as
English	A cannabinoid receptor 1 mutation proximal to the DRY motif results in constitutive activity and reveals intramolecular interactions involved in receptor activation	scientific article published on 31 July 2006

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scholarly article

1 reference

Europe PubMed Central

19 August 2017

A cannabinoid receptor 1 mutation proximal to the DRY motif results in constitutive activity and reveals intramolecular interactions involved in receptor activation (English)

1 reference

Europe PubMed Central

19 August 2017

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cannabinoid receptor

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author name string

Aaron M D'Antona

1

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Europe PubMed Central

19 August 2017

Kwang H Ahn

2

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Europe PubMed Central

19 August 2017

Lei Wang

3

1 reference

Europe PubMed Central

19 August 2017

Dale F Mierke

4

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Europe PubMed Central

19 August 2017

Jean Lucas-Lenard

5

1 reference

Europe PubMed Central

19 August 2017

Debra A Kendall

6

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Europe PubMed Central

19 August 2017

language of work or name

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publication date

31 July 2006

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Europe PubMed Central

19 August 2017

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Europe PubMed Central

19 August 2017

1108

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Europe PubMed Central

19 August 2017

1

1 reference

Europe PubMed Central

19 August 2017

1-11

1 reference

Europe PubMed Central

19 August 2017

Mutations of CB1 T210 produce active and inactive receptor forms: correlations with ligand affinity, receptor stability, and cellular localization

1 reference

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6 September 2017

Efficacy in CB1 receptor-mediated signal transduction

1 reference

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An Aromatic Microdomain at the Cannabinoid CB1 Receptor Constitutes an Agonist/Inverse Agonist Binding Region

1 reference

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6 September 2017

GPCRDB information system for G protein-coupled receptors

1 reference

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International Union of Pharmacology. XXVII. Classification of cannabinoid receptors

1 reference

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Endocannabinoid signaling in the brain

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Crystal structure of rhodopsin: A G protein-coupled receptor

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Uncovering molecular mechanisms involved in activation of G protein-coupled receptors

1 reference

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C5a receptor activation. Genetic identification of critical residues in four transmembrane helices

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Constitutive activation of a single effector pathway: evidence for multiple activation states of a G protein-coupled receptor.

1 reference

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1 reference

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A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

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Chemically distinct ligands promote differential CB1 cannabinoid receptor-Gi protein interactions.

1 reference

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Structural mimicry in class A G protein-coupled receptor rotamer toggle switches: the importance of the F3.36(201)/W6.48(357) interaction in cannabinoid CB1 receptor activation

1 reference

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Activation of the beta 2-adrenergic receptor involves disruption of an ionic lock between the cytoplasmic ends of transmembrane segments 3 and 6.

1 reference

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Constitutive precoupling to G(i) and increased agonist potency in the alpha(2B)-adrenoceptor

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Mutational analysis of the highly conserved arginine within the Glu/Asp-Arg-Tyr motif of the alpha(1b)-adrenergic receptor: effects on receptor isomerization and activation.

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1 reference

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Ligand binding and modulation of cyclic AMP levels depend on the chemical nature of residue 192 of the human cannabinoid receptor 1.

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Identifiers

10.1016/J.BRAINRES.2006.05.042

1 reference

Europe PubMed Central

19 August 2017

1 reference

Europe PubMed Central

19 August 2017

1 reference

Europe PubMed Central

19 August 2017

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