Discriminative stimulus functions in rats of AM1346, a high-affinity CB1R selective anandamide analog (Q37055254)

18 August 2017

Discriminative stimulus functions in rats of AM1346, a high-affinity CB1R selective anandamide analog (English)

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18 August 2017

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Alexandros Makriyannis

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4

object named as

Alexandros Makriyannis

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18 August 2017

Torbjörn U C Järbe

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PMCID

3727224

18 August 2017

Chen Li

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2

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PMCID

3727224

18 August 2017

Qian Liu

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3

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18 August 2017

3 June 2008

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18 August 2017

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18 August 2017

203

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18 August 2017

229-239

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18 August 2017

2

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https://scigraph.springernature.com/pub.10.1007/s00213-008-1199-3

18 August 2017

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29 September 2017

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29 September 2017

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A comparison of the discriminative stimulus effects of delta(9)-tetrahydrocannabinol and O-1812, a potent and metabolically stable anandamide analog, in rats

29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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Unique agonist-bound cannabinoid CB1 receptor conformations indicate agonist specificity in signaling

29 September 2017

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Effects of AM1346, a high-affinity CB1 receptor selective anandamide analog, on open-field behavior in rats

27 June 2018

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The cannabinoid receptor antagonist SR-141716 does not readily antagonize open-field effects induced by the cannabinoid receptor agonist (R)-methanandamide in rats

27 June 2018

1 reference

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Effects of delta-9-tetrahydrocannabinol and (R)-methanandamide on open-field behavior in rats.

27 June 2018

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Delta9-THC training dose as a determinant for (R)-methanandamide generalization in rats.

27 June 2018

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Novel analogues of arachidonylethanolamide (anandamide): affinities for the CB1 and CB2 cannabinoid receptors and metabolic stability.

27 June 2018

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A repeated test procedure to assess onset and duration of the cue properties of (-) delta 9-THC, (-) delta 8-THC-DMH and (+) delta 8-THC.

27 June 2018

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Discriminative Stimulus Properties of Δ9-Tetrahydrocannabinol: Mechanistic Studies

27 June 2018

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Cannabimimetic activity (delta 1-THC cue) of cannabidiol monomethyl ether and two stereoisomeric hexahydrocannabinols in rats and pigeons.

27 June 2018

1 reference

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A comparison of the discriminative stimulus properties of delta 9-tetrahydrocannabinol and CP 55,940 in rats and rhesus monkeys

27 June 2018

1 reference

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Delta9-THC training dose as a determinant for (R)-methanandamide generalization in rats: a systematic replication.

27 June 2018

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The endogenous cannabinoid anandamide produces delta-9-tetrahydrocannabinol-like discriminative and neurochemical effects that are enhanced by inhibition of fatty acid amide hydrolase but not by inhibition of anandamide transport.

21 January 2018

1 reference

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Discriminative stimulus functions of AM-1346, a CB1R selective anandamide analog in rats trained with Delta9-THC or (R)-methanandamide (AM-356).

4 September 2018

1 reference

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Characterization of cannabinoid agonists and apparent pA2 analysis of cannabinoid antagonists in rhesus monkeys discriminating Delta9-tetrahydrocannabinol.

4 September 2018

1 reference

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(-)-7'-Isothiocyanato-11-hydroxy-1',1'-dimethylheptylhexahydrocannabinol (AM841), a high-affinity electrophilic ligand, interacts covalently with a cysteine in helix six and activates the CB1 cannabinoid receptor

4 September 2018

1 reference

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Increasing the selectivity of the discriminative stimulus effects of delta 9-tetrahydrocannabinol: complete substitution with methanandamide

4 September 2018

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(R)-Methanandamide and delta9-tetrahydrocannabinol-induced operant rate decreases in rats are not readily antagonized by SR-141716A.

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3727224

Inhibition of methamphetamine self-administration in rats by cannabinoid receptor antagonist AM 251.

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3727224

(R)-methanandamide and Delta 9-THC as discriminative stimuli in rats: tests with the cannabinoid antagonist SR-141716 and the endogenous ligand anandamide

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3727224

Dual activation and inhibition of adenylyl cyclase by cannabinoid receptor agonists: evidence for agonist-specific trafficking of intracellular responses.

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3727224

Differential receptor-G-protein coupling evoked by dissimilar cannabinoid receptor agonists.

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3727224

Evaluation of cannabimimetic effects of structural analogs of anandamide in rats

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3727224

(R)-methanandamide, but not anandamide, substitutes for delta 9-THC in a drug-discrimination procedure.

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3727224

Pharmacological specificity of delta 9-tetrahydrocannabinol discrimination in rats

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3727224

Inter-animal olfactory cues in operant drug discrimination procedures in rats.

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3727224

WIN55212-2 docking to the CB1 cannabinoid receptor and multiple pathways for conformational induction

4 September 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/18521574

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1007/S00213-008-1199-3

1 reference

18 August 2017

1 reference

18 August 2017

1 reference

PMCID

3727224