URB602 inhibits monoacylglycerol lipase and selectively blocks 2-arachidonoylglycerol degradation in intact brain slices. (Q36427265)

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30 December 2019

title

URB602 inhibits monoacylglycerol lipase and selectively blocks 2-arachidonoylglycerol degradation in intact brain slices (English)

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30 December 2019

main subject

glyceryl 2-arachidonate

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author

Silvia Rivara

4

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30 December 2019

Giuseppe Astarita

7

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30 December 2019

Marco Mor

10

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30 December 2019

2

Andrea Duranti

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30 December 2019

3

Andrea Tontini

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30 December 2019

11

Giorgio Tarzia

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30 December 2019

6

Jason R Clapper

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30 December 2019

author name string

Alvin R King

1

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30 December 2019

Anja Rosengarth

5

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30 December 2019

Jennifer A Geaga

8

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Hartmut Luecke

9

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Daniele Piomelli

12

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publication date

1 December 2007

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30 December 2019

published in

Chemistry and Biology

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volume

14

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issue

12

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30 December 2019

page(s)

1357-1365

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The inhibition of monoacylglycerol lipase by URB602 showed an anti-inflammatory and anti-nociceptive effect in a murine model of acute inflammation

30 December 2019

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URB754 has no effect on the hydrolysis or signaling capacity of 2-AG in the rat brain

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30 September 2017

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cDNA cloning, tissue distribution, and identification of the catalytic triad of monoglyceride lipase. Evolutionary relationship to esterases, lysophospholipases, and haloperoxidases

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30 September 2017

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30 September 2017

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Molecular characterization of an enzyme that degrades neuromodulatory fatty-acid amides

30 September 2017

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Irreversible inhibition of Ca(2+)-independent phospholipase A2 by methyl arachidonyl fluorophosphonate

30 September 2017

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30 September 2017

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30 September 2017

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21 September 2018

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21 September 2018

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21 September 2018

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10.1016/J.CHEMBIOL.2007.10.017

21 September 2018

Identifiers

DOI

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