Biochemical and pharmacological profile of a potent and selective endothelin B-receptor antagonist, BQ-788. (Q35315000)

7 August 2017

Biochemical and pharmacological profile of a potent and selective endothelin B-receptor antagonist, BQ-788. (English)

1 reference

7 August 2017

K Ishikawa

1

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7 August 2017

M Ihara

2

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7 August 2017

K Noguchi

3

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7 August 2017

T Mase

4

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7 August 2017

N Mino

5

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7 August 2017

T Saeki

6

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7 August 2017

T Fukuroda

7

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7 August 2017

T Fukami

8

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7 August 2017

S Ozaki

9

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7 August 2017

T Nagase

10

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7 August 2017

language of work or name

English

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publication date

1 May 1994

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Proceedings of the National Academy of Sciences of the United States of America

7 August 2017

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7 August 2017

91

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7 August 2017

11

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7 August 2017

4892-4896

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A novel ETA-receptor antagonist, FR 139317, inhibits endothelin-induced contractions of guinea-pig pulmonary arteries, but not trachea

7 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

A new generation of Ca2+ indicators with greatly improved fluorescence properties

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Autoradiographic distribution in rat tissues of binding sites for endothelin: a neuropeptide?

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

The human endothelin family: three structurally and pharmacologically distinct isopeptides predicted by three separate genes

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

A novel potent vasoconstrictor peptide produced by vascular endothelial cells

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Cloning of a cDNA encoding a non-isopeptide-selective subtype of the endothelin receptor

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Cloning and expression of a cDNA encoding an endothelin receptor

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Endothelin receptor subtypes and stimulation of aldosterone secretion

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Cloning and functional expression of a vascular smooth muscle endothelin 1 receptor

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Two endothelin receptor subtypes in porcine arteries.

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Cloning and sequence analysis of a cDNA encoding human non-selective type of endothelin receptor

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Primary structure of bovine endothelin ETB receptor and identification of signal peptidase and metal proteinase cleavage sites

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

[Ala1,3,11,15]endothelin-1 analogs with ETB agonistic activity.

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Cloning and expression of human endothelin-1 receptor cDNA

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Molecular cloning of a non-isopeptide-selective human endothelin receptor

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

BQ-123, cyclo(-D-Trp-D-Asp-Pro-D-Val-Leu), is a non-competitive antagonist of the actions of endothelin-1 in SK-N-MC human neuroblastoma cells

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Pharmacological evidence for distinct endothelin receptors in guinea-pig bronchus and aorta

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

A novel radioligand [125I]BQ-3020 selective for endothelin (ETB) receptors

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Cyclic pentapeptide endothelin antagonists with high ETA selectivity. Potency- and solubility-enhancing modifications

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Molecular cloning and characterization of the major endothelin receptor subtype in porcine cerebellum

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Biological profiles of highly potent novel endothelin antagonists selective for the ETA receptor

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Non-isopeptide-selective endothelin receptors in human girardi heart cells

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

An endothelin B receptor-selective antagonist: IRL 1038, [Cys11-Cys15]-endothelin-1(11-21)

27 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=43895

Antihypertensive effect of a newly synthesized endothelin antagonist, BQ-123, in a genetic hypertensive model

26 September 2018

1 reference

12 December 2020

Role of endothelin ETB receptors in bronchoconstrictor and vasoconstrictor responses in guinea-pigs

1 reference

12 December 2020

Interaction of circulating cell-derived and plasma growth factors in stimulating cultured smooth muscle cell replication

1 reference

12 December 2020

Autoradiographic visualization of the binding sites for [125I]endothelin in rat and human brain

1 reference

12 December 2020

Presence of non-selective type of endothelin receptor on vascular endothelium and its linkage to vasodilation

1 reference

12 December 2020

Endothelin and structurally related analogs distinguish between endothelin receptor subtypes

1 reference

12 December 2020

Analysis of responses to endothelins in isolated porcine blood vessels by using a novel endothelin antagonist, BQ-153

1 reference

12 December 2020

Venous smooth muscle contains vasoconstrictor ETB-like receptors

1 reference

12 December 2020

Identifiers

DOI

10.1073/PNAS.91.11.4892

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7 August 2017

0 references

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7 August 2017

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