Efficacy at G-protein-coupled receptors (Q34742798)

4 August 2017

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title

Efficacy at G-protein-coupled receptors (English)

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G protein-coupled receptor

4 August 2017

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author name string

Terry Kenakin

series ordinal

1

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4 August 2017

1 February 2002

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Nature Reviews Drug Discovery

4 August 2017

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4 August 2017

1

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4 August 2017

103-110

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4 August 2017

2

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https://scigraph.springernature.com/pub.10.1038/nrd722

4 August 2017

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Treatment with inverse agonists enhances baseline atrial contractility in transgenic mice with chronic beta2-adrenoceptor activation

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31 March 2020

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Creation and functional screening of a multi-use peptide library

31 March 2020

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Tools for investigating functional interactions between ligands and G-protein-coupled receptors

31 March 2020

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The cubic ternary complex receptor-occupancy model. III. resurrecting efficacy

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Can allosteric regulation be predicted from structure?

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Energetics of Ligand Binding to Proteins

31 March 2020

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inferred from DOI database lookup

7 January 2021

based on heuristic

Hydrogen Exchange in Proteins

1 reference

inferred from DOI database lookup

7 January 2021

based on heuristic

Recombinant human CXC-chemokine receptor-4 in melanophores are linked to Gi protein: seven transmembrane coreceptors for human immunodeficiency virus entry into cells

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inferred from DOI database lookup

7 January 2021

based on heuristic

Identifiers

DOI

10.1038/NRD722

1 reference

4 August 2017

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PubMed ID

12120091