Inhibitors of human heart chymase based on a peptide library (Q34074276)

30 July 2017

Inhibitors of human heart chymase based on a peptide library (English)

1 reference

30 July 2017

3

R H Abeles

1 reference

30 July 2017

M Bastos

1

1 reference

PubMed ID

7624313

30 July 2017

N J Maeji

series ordinal

2

1 reference

PubMed ID

7624313

30 July 2017

language of work or name

English

0 references

publication date

1 July 1995

1 reference

Proceedings of the National Academy of Sciences of the United States of America

30 July 2017

1 reference

30 July 2017

92

1 reference

30 July 2017

15

1 reference

30 July 2017

6738-6742

1 reference

On the attribution and additivity of binding energies

30 July 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

Mapping the S' subsites of serine proteases using acyl transfer to mixtures of peptide nucleophiles

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

Identification of substrate-analog trypsin inhibitors through the screening of synthetic peptide combinatorial libraries

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

Applications of combinatorial technologies to drug discovery. 1. Background and peptide combinatorial libraries

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

Creation and functional screening of a multi-use peptide library

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

Use of synthetic peptide libraries and phosphopeptide-selective mass spectrometry to probe protein kinase substrate specificity.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

Phosphonamidates as transition-state analogue inhibitors of thermolysin.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

On the size of the active site in proteases. I. Papain

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

Mechanism of slow-binding inhibition of human leukocyte elastase by trifluoromethyl ketones.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

Inhibition of cathepsin B and papain by peptidyl alpha-keto esters, alpha-keto amides, alpha-diketones, and alpha-keto acids

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

Structure-activity studies of fluoroketone inhibitors of alpha-lytic protease and human leukocyte elastase

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

Multiple determinants for the high substrate specificity of an angiotensin II-forming chymase from the human heart

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

.alpha.-Keto amide inhibitors of aminopeptidases

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

Rapid optimization of enzyme substrates using defined substrate mixtures

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

Reaction of peptide aldehydes with serine proteases. Implications for the entropy changes associated with enzymic catalysis

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

A new type of synthetic peptide library for identifying ligand-binding activity

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=41404

Inhibition of chymotrypsin by fluorinated alpha-keto acid derivatives

28 October 2018

1 reference

12 December 2020

Alpha-diketone and alpha-keto ester derivatives of N-protected amino acids and peptides as novel inhibitors of cysteine and serine proteinases

1 reference

12 December 2020

Peptide alpha-keto ester, alpha-keto amide, and alpha-keto acid inhibitors of calpains and other cysteine proteases

1 reference

12 December 2020

Angiotensin II-forming pathways in normal and failing human hearts

1 reference

12 December 2020

Stereospecific synthesis of peptidyl alpha-keto amides as inhibitors of calpain

1 reference

12 December 2020

Inactivation of calpain by peptidyl fluoromethyl ketones

1 reference

12 December 2020

The rapid identification of HIV protease inhibitors through the synthesis and screening of defined peptide mixtures

1 reference

12 December 2020

Extended binding inhibitors of chymotrypsin that interact with leaving group subsites S1'-S3'

1 reference

12 December 2020

Synthesis of peptidyl fluoromethyl ketones and peptidyl alpha-keto esters as inhibitors of porcine pancreatic elastase, human neutrophil elastase, and rat and human neutrophil cathepsin G

1 reference

12 December 2020

Tight-binding inhibitors-I. Kinetic behavior

1 reference

12 December 2020

Identifiers

DOI

10.1073/PNAS.92.15.6738

1 reference

30 July 2017

0 references

1 reference

30 July 2017

1 reference

PubMed ID

7624313