Fluorinated cannabinoid CB2 receptor ligands: synthesis and in vitro binding characteristics of 2-oxoquinoline derivatives (Q34004234)

30 July 2017

Fluorinated cannabinoid CB2 receptor ligands: synthesis and in vitro binding characteristics of 2-oxoquinoline derivatives (English)

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30 July 2017

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Nashaat Turkman

1

1 reference

30 July 2017

Aleksander Shavrin

2

1 reference

30 July 2017

Roman A Ivanov

3

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30 July 2017

Brian Rabinovich

4

1 reference

30 July 2017

Andrei Volgin

5

1 reference

30 July 2017

Juri G Gelovani

6

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30 July 2017

Mian M Alauddin

7

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30 July 2017

language of work or name

English

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publication date

5 August 2011

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Bioorganic & Medicinal Chemistry

30 July 2017

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30 July 2017

19

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30 July 2017

18

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30 July 2017

5698-5707

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Synthesis and in vitro biological evaluation of carbon-11-labeled quinoline derivatives as new candidate PET radioligands for cannabinoid CB2 receptor imaging

30 July 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3174488

Synthetic cannabinoid receptor agonists inhibit tumor growth and metastasis of breast cancer

28 July 2018

1 reference

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The cannabinoid CB2 receptor as a target for inflammation-dependent neurodegeneration

28 July 2018

1 reference

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Sulfamoyl benzamides as novel CB2 cannabinoid receptor ligands

28 July 2018

1 reference

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Recent advances in the development of selective ligands for the cannabinoid CB(2) receptor

28 July 2018

1 reference

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Cannabinoid receptor agonist-induced apoptosis of human prostate cancer cells LNCaP proceeds through sustained activation of ERK1/2 leading to G1 cell cycle arrest

28 July 2018

1 reference

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Endocannabinoids and the gastrointestinal tract

28 July 2018

1 reference

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Design, synthesis, and binding studies of new potent ligands of cannabinoid receptors

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3174488

28 July 2018

1 reference

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Recent developments in the medicinal chemistry of cannabimimetic indoles, pyrroles and indenes

28 July 2018

1 reference

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Prevention of Alzheimer's disease pathology by cannabinoids: neuroprotection mediated by blockade of microglial activation.

28 July 2018

1 reference

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C-3 Amido-indole cannabinoid receptor modulators

28 July 2018

1 reference

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International Union of Pharmacology. XXVII. Classification of cannabinoid receptors

28 July 2018

1 reference

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Antiinflammatory action of endocannabinoid palmitoylethanolamide and the synthetic cannabinoid nabilone in a model of acute inflammation in the rat

28 July 2018

1 reference

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Functional role of tryptophan residues in the fourth transmembrane domain of the CB(2) cannabinoid receptor

28 July 2018

1 reference

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3-(1',1'-Dimethylbutyl)-1-deoxy-delta8-THC and related compounds: synthesis of selective ligands for the CB2 receptor

28 July 2018

1 reference

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Cannabinoid receptor interactions with the antagonists SR 141716A and SR 144528.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3174488

Structure-activity relationships of indole- and pyrrole-derived cannabinoids

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3174488

SR 144528, the first potent and selective antagonist of the CB2 cannabinoid receptor.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3174488

Evaluation of binding in a transfected cell line expressing a peripheral cannabinoid receptor (CB2): identification of cannabinoid receptor subtype selective ligands.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3174488

Molecular characterization of a peripheral receptor for cannabinoids

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3174488

Comparison of the pharmacology and signal transduction of the human cannabinoid CB1 and CB2 receptors

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3174488

Synthesis and biological evaluation of carbon-11- and fluorine-18-labeled 2-oxoquinoline derivatives for type 2 cannabinoid receptor positron emission tomography imaging.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3174488

"Click labeling" with 2-[18f]fluoroethylazide for positron emission tomography.

29 October 2018

1 reference

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Cannabinoid receptors as novel targets for the treatment of melanoma

29 October 2018

1 reference

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Synthesis and SAR studies of 2-oxoquinoline derivatives as CB2 receptor inverse agonists.

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3174488

Virtual screening of novel CB2 ligands using a comparative model of the human cannabinoid CB2 receptor.

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3174488

A novel cannabinoid peripheral cannabinoid receptor-selective inverse agonist blocks leukocyte recruitment in vivo

29 October 2018

1 reference

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Current knowledge on the antagonists and inverse agonists of cannabinoid receptors.

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3174488

Targeting the cannabinoid CB2 receptor: mutations, modeling and development of CB2 selective ligands.

29 October 2018

1 reference

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Inflammation and autoimmunity as a central theme in neurodegenerative disorders: fact or fiction?

29 October 2018

1 reference

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Tricyclic pyrazoles. Part 1: synthesis and biological evaluation of novel 1,4-dihydroindeno[1,2-c]pyrazol-based ligands for CB1and CB2 cannabinoid receptors.

29 October 2018

1 reference

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1-Methoxy-, 1-deoxy-11-hydroxy- and 11-hydroxy-1-methoxy-Delta(8)-tetrahydrocannabinols: new selective ligands for the CB2 receptor

29 October 2018

1 reference

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Resorcinol derivatives: a novel template for the development of cannabinoid CB(1)/CB(2) and CB(2)-selective agonists

29 October 2018

1 reference

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In vitro and in vivo pharmacological characterization of JTE-907, a novel selective ligand for cannabinoid CB2 receptor

29 October 2018

1 reference

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SR141716A, a potent and selective antagonist of the brain cannabinoid receptor

29 October 2018

1 reference

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Synthesis and in vitro evaluation of novel 2-oxo-1,2-dihydroquinoline CB2 receptor inverse agonists

29 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21872477

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Effects of cannabinoid receptor ligands on LPS-induced pulmonary inflammation in mice

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21872477

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Overexpression of cannabinoid receptors CB1 and CB2 correlates with improved prognosis of patients with hepatocellular carcinoma

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21872477

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.BMC.2011.07.062

1 reference

30 July 2017

1 reference

30 July 2017

1 reference