Synthesis and positron emission tomography studies of carbon-11-labeled imatinib (Gleevec). (Q33836021)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17307123%20AND%20SRC:MED&resulttype=core&format=json

25 December 2019

title

Synthesis and positron emission tomography studies of carbon-11-labeled imatinib (Gleevec) (English)

1 reference

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positron emission tomography

25 December 2019

main subject

1 reference

1 reference

3

1 reference

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25 December 2019

9

Joanna S Fowler

1 reference

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25 December 2019

author name string

Kun-Eek Kil

1

1 reference

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25 December 2019

Yu-Shin Ding

2

1 reference

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25 December 2019

David Alexoff

4

1 reference

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25 December 2019

Sung Won Kim

5

1 reference

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25 December 2019

Colleen Shea

6

1 reference

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25 December 2019

Youwen Xu

7

1 reference

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25 December 2019

Lisa Muench

8

1 reference

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25 December 2019

publication date

1 February 2007

1 reference

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Nuclear Medicine and Biology

25 December 2019

published in

1 reference

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25 December 2019

volume

34

1 reference

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25 December 2019

issue

2

1 reference

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25 December 2019

page(s)

153-163

1 reference

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Cardiotoxicity of the cancer therapeutic agent imatinib mesylate.

25 December 2019

cites work

1 reference

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Comparative evaluation of positron emission tomography radiotracers for imaging the norepinephrine transporter: (S,S) and (R,R) enantiomers of reboxetine analogs ([11C]methylreboxetine, 3-Cl-[11C]methylreboxetine and [18F]fluororeboxetine), (R)-[11C

4 July 2018

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Inhibition of platelet-derived growth factor signaling attenuates pulmonary fibrosis.

4 July 2018

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Rational approaches to the design of therapeutics targeting molecular markers: the case of chronic myelogenous leukemia

4 July 2018

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The development of imatinib as a therapeutic agent for chronic myeloid leukemia

4 July 2018

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Progression-free survival in gastrointestinal stromal tumours with high-dose imatinib: randomised trial

4 July 2018

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Imatinib (STI571) resistance in chronic myelogenous leukemia: molecular basis of the underlying mechanisms and potential strategies for treatment

4 July 2018

1 reference

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Gleevec inhibits β-amyloid production but not Notch cleavage

4 July 2018

1 reference

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Specific targeted therapy of chronic myelogenous leukemia with imatinib

4 July 2018

1 reference

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Distribution of STI-571 to the brain is limited by P-glycoprotein-mediated efflux

4 July 2018

1 reference

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Activity of the Bcr-Abl kinase inhibitor PD180970 against clinically relevant Bcr-Abl isoforms that cause resistance to imatinib mesylate (Gleevec, STI571).

4 July 2018

1 reference

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Crystal structures of the kinase domain of c-Abl in complex with the small molecule inhibitors PD173955 and imatinib (STI-571)

4 July 2018

1 reference

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Protein kinases--the major drug targets of the twenty-first century?

4 July 2018

1 reference

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Approval summary for imatinib mesylate capsules in the treatment of chronic myelogenous leukemia.

4 July 2018

1 reference

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STI571 inactivation of the gastrointestinal stromal tumor c-KIT oncoprotein: biological and clinical implications

4 July 2018

1 reference

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Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings

4 July 2018

1 reference

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Abl protein-tyrosine kinase inhibitor STI571 inhibits in vitro signal transduction mediated by c-kit and platelet-derived growth factor receptors

4 July 2018

1 reference

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Selection and characterization of BCR-ABL positive cell lines with differential sensitivity to the tyrosine kinase inhibitor STI571: diverse mechanisms of resistance.

4 July 2018

1 reference

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KIT extracellular and kinase domain mutations in gastrointestinal stromal tumors

4 July 2018

1 reference

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PET and drug research and development

4 July 2018

1 reference

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Gastrointestinal pacemaker cell tumor (GIPACT): gastrointestinal stromal tumors show phenotypic characteristics of the interstitial cells of Cajal

4 July 2018

1 reference

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Gain-of-function mutations of c-kit in human gastrointestinal stromal tumors

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2866181

Synthesis and in vivo evaluation of a 99m/99Tc-DADT-benzovesamicol: a potential marker for cholinergic neurons.

4 July 2018

1 reference

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Effects of a selective inhibitor of the Abl tyrosine kinase on the growth of Bcr-Abl positive cells

4 July 2018

1 reference

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Letter: A new consistent chromosomal abnormality in chronic myelogenous leukaemia identified by quinacrine fluorescence and Giemsa staining

4 July 2018

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F-18 FDG PET for assessing tyrosine kinase-related signal transduction inhibition in a GIST c-kit-positive tumor patient by imatinib.

4 July 2018

1 reference

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Oral imatinib treatment reduces early fibrogenesis but does not prevent progression in the long term.

29 October 2018

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Imatinib as a novel antifibrotic agent in bleomycin-induced pulmonary fibrosis in mice

29 October 2018

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Imatinib mesylate (STI-571) attenuates liver fibrosis development in rats.

29 October 2018

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Successful treatment of hepatocellular carcinoma with the tyrosine kinase inhibitor imatinib in a patient with liver cirrhosis

29 October 2018

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Absolute bioavailability of imatinib (Glivec) orally versus intravenous infusion

29 October 2018

1 reference

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Association of KIT exon 9 mutations with nongastric primary site and aggressive behavior: KIT mutation analysis and clinical correlates of 120 gastrointestinal stromal tumors

29 October 2018

1 reference

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Imatinib mesylate has limited activity against the central nervous system involvement of Philadelphia chromosome-positive acute lymphoblastic leukaemia due to poor penetration into cerebrospinal fluid

29 October 2018

1 reference

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Treatment of inoperable gastrointestinal stromal tumor (GIST) with Imatinib (Glivec, Gleevec).

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2866181

Carbon-11-d-threo-methylphenidate binding to dopamine transporter in baboon brain

29 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/17307123

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

The tyrosine kinase inhibitor CGP57148B selectively inhibits the growth of BCR-ABL-positive cells

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/17307123

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

The effect of Bcrp1 (Abcg2) on the in vivo pharmacokinetics and brain penetration of imatinib mesylate (Gleevec): implications for the use of breast cancer resistance protein and P-glycoprotein inhibitors to enable the brain penetration of imatinib

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/17307123

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.NUCMEDBIO.2006.11.004

1 reference

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25 December 2019

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17307123%20AND%20SRC:MED&resulttype=core&format=json

25 December 2019

1 reference