Persistent activation by and receptor reserve for an irreversible A1-adenosine receptor agonist in DDT1 MF-2 cells and in guinea pig heart (Q33802589)

29 July 2017

title

Persistent activation by and receptor reserve for an irreversible A1-adenosine receptor agonist in DDT1 MF-2 cells and in guinea pig heart (English)

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29 July 2017

J Zhang

1

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29 July 2017

L Belardinelli

2

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29 July 2017

K A Jacobson

3

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29 July 2017

D H Otero

4

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29 July 2017

S P Baker

5

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29 July 2017

publication date

1 September 1997

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29 July 2017

published in

Molecular Pharmacology

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29 July 2017

volume

52

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29 July 2017

issue

3

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29 July 2017

page(s)

491-498

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A modification of receptor theory

29 July 2017

cites work

1 reference

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An irreversible A1-selective adenosine agonist preconditions rabbit heart.

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1,3-Dipropyl-8-[2-(5,6-epoxy)norbornyl]xanthine, a potent, specific and selective A1 adenosine receptor antagonist in the guinea pig heart and brain and in DDT1MF-2 cells.

28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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Distinct pathways of desensitization of A1- and A2-adenosine receptors in DDT1 MF-2 cells

28 July 2018

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28 July 2018

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Evidence of spare A1-adenosine receptors in guinea pig atrioventricular node

28 July 2018

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28 July 2018

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Adenosine A1-receptor stimulation of inositol phospholipid hydrolysis and calcium mobilisation in DDT1 MF-2 cells

28 July 2018

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28 July 2018

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28 July 2018

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Differential effects of alkylating agents on the multiple muscarinic receptor subtypes linked to activation of phospholipase C by carbachol in rat brain cortical membranes

28 July 2018

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Differences in muscarinic receptor reserve for inhibition of adenylate cyclase and stimulation of phosphoinositide hydrolysis in chick heart cells

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12 December 2020

Mechanism of A2 adenosine receptor activation. I. Blockade of A2 adenosine receptors by photoaffinity labeling

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12 December 2020

Biochemical and physical analyses of newly synthesized muscarinic acetylcholine receptors in cultured embryonic chicken cardiac cells

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12 December 2020

Substituted 1,3-dipropylxanthines as irreversible antagonists of A1 adenosine receptors.

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12 December 2020

Characterization of adenosine receptors in the PC12 pheochromocytoma cell line using radioligand binding: evidence for A-2 selectivity

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12 December 2020

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12 December 2020

G protein-dependent activation of phospholipase C by adenosine A3 receptors in rat brain

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12 December 2020

Propylbenzilylcholine mustard labels an acidic residue in transmembrane helix 3 of the muscarinic receptor

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12 December 2020

Identifiers

PMC publication ID

5472056

1 reference

29 July 2017

1 reference