Identification of broad-based HIV-1 protease inhibitors from combinatorial libraries (Q33589171)

28 July 2017

title

Identification of broad-based HIV-1 protease inhibitors from combinatorial libraries (English)

1 reference

28 July 2017

Max W Chang

1

0 references

Sukwon Hong

object named as

Sukwon Hong

6

0 references

author name string

Michael J Giffin

2

1 reference

28 July 2017

Rolf Muller

3

1 reference

28 July 2017

Jeremiah Savage

4

1 reference

28 July 2017

Ying C Lin

5

1 reference

28 July 2017

Wei Jin

7

1 reference

28 July 2017

Landon R Whitby

8

1 reference

28 July 2017

John H Elder

9

1 reference

28 July 2017

Dale L Boger

10

1 reference

28 July 2017

Bruce E Torbett

11

1 reference

28 July 2017

language of work or name

English

0 references

publication date

1 August 2010

1 reference

28 July 2017

number of pages

6

1 reference

based on heuristic

inferred from page(s)

published in

Biochemical Journal

1 reference

28 July 2017

volume

429

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28 July 2017

issue

3

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28 July 2017

page(s)

527-532

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Fragment-Based Screen against HIV Protease

28 July 2017

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Discovery of inhibitors of aberrant gene transcription from Libraries of DNA binding molecules: inhibition of LEF-1-mediated gene transcription and oncogenic transformation

21 June 2018

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Viral protease inhibitors

21 June 2018

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A copper(I)-catalyzed 1,2,3-triazole azide-alkyne click compound is a potent inhibitor of a multidrug-resistant HIV-1 protease variant

21 June 2018

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Solution kinetics measurements suggest HIV-1 protease has two binding sites for darunavir and amprenavir

21 June 2018

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Targeting the open-flap conformation of HIV-1 protease with pyrrolidine-based inhibitors

21 June 2018

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21 June 2018

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A poke in the eye: inhibiting HIV-1 protease through its flap-recognition pocket

21 June 2018

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HIV-1 protease folding and the design of drugs which do not create resistance

21 June 2018

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21 June 2018

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21 June 2018

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Beta-lactam compounds as apparently uncompetitive inhibitors of HIV-1 protease

21 June 2018

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Development of low molecular weight HIV-1 protease dimerization inhibitors

21 June 2018

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HIV-1 protease molecular dynamics of a wild-type and of the V82F/I84V mutant: possible contributions to drug resistance and a potential new target site for drugs

21 June 2018

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Solution‐Phase Combinatorial Libraries: Modulating Cellular Signaling by Targeting Protein–Protein or Protein–DNA Interactions

21 June 2018

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21 June 2018

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A Common Mechanism Underlying Promiscuous Inhibitors from Virtual and High-Throughput Screening

21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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Human immunodeficiency virus has an aspartic-type protease that can be inhibited by pepstatin A

21 June 2018

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Stability and activity of human immunodeficiency virus protease: comparison of the natural dimer with a homologous, single-chain tethered dimer

21 June 2018

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Crystallographic analysis of a complex between human immunodeficiency virus type 1 protease and acetyl-pepstatin at 2.0-A resolution

21 June 2018

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A simple, continuous fluorometric assay for HIV protease

21 June 2018

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Switching between allosteric and dimerization inhibition of HIV-1 protease

21 June 2018

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https://api.crossref.org/works/10.1042%2FBJ20091645

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Analysis of the combined effect of two linear inhibitors on a single enzyme

21 January 2018

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Synergistic binding of inhibitors to the protease from HIV type 1.

31 October 2018

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STUDIES ON LIVER ALCOHOL HYDROGENASE COMPLEXES. 3. MULTIPLE INHIBITION KINETICS IN THE PRESENCE OF TWO COMPETITIVE INHIBITORS

31 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20507280

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12 December 2020

based on heuristic

Evaluation of enzyme inhibitors in drug discovery. A guide for medicinal chemists and pharmacologists

1 reference

PubMed

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inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1042/BJ20091645

1 reference

28 July 2017

1 reference

28 July 2017

1 reference