Structure-based development of novel adenylyl cyclase inhibitors (Q33352228)

26 July 2017

title

Structure-based development of novel adenylyl cyclase inhibitors (English)

1 reference

26 July 2017

Lonny R Levin

5

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Jochen Buck

6

object named as

Jochen Buck

1 reference

26 July 2017

7

Clemens Steegborn

1 reference

26 July 2017

Christine Schlicker

1

1 reference

26 July 2017

Annika Rauch

2

1 reference

26 July 2017

Ken C Hess

3

1 reference

26 July 2017

Barbara Kachholz

4

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26 July 2017

language of work or name

English

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publication date

17 July 2008

1 reference

Journal of Medicinal Chemistry

26 July 2017

published in

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26 July 2017

volume

51

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26 July 2017

issue

15

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26 July 2017

page(s)

4456-4464

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Activation and inhibition of adenylyl cyclase isoforms by forskolin analogs.

26 July 2017

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Drug therapy aimed at adenylyl cyclase to regulate cyclic nucleotide signaling

28 July 2018

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The "soluble" adenylyl cyclase in sperm mediates multiple signaling events required for fertilization

28 July 2018

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A novel mechanism for adenylyl cyclase inhibition from the crystal structure of its complex with catechol estrogen

28 July 2018

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Bicarbonate activation of adenylyl cyclase via promotion of catalytic active site closure and metal recruitment

28 July 2018

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Virtual screening of human 5-aminoimidazole-4-carboxamide ribonucleotide transformylase against the NCI diversity set by use of AutoDock to identify novel nonfolate inhibitors

28 July 2018

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Tyrphostins are inhibitors of guanylyl and adenylyl cyclases

28 July 2018

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28 July 2018

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Differential inhibition of adenylyl cyclase isoforms and soluble guanylyl cyclase by purine and pyrimidine nucleotides.

28 July 2018

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The class III adenylyl cyclases: multi-purpose signalling modules

28 July 2018

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Bicarbonate-regulated Adenylyl Cyclase (sAC) Is a Sensor That Regulates pH-dependent V-ATPase Recycling

28 July 2018

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Metal Coordination-Based Inhibitors of Adenylyl Cyclase: Novel Potent P-Site Antagonists

28 July 2018

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Isoform-targeted regulation of cardiac adenylyl cyclase.

28 July 2018

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Kinetic properties of "soluble" adenylyl cyclase. Synergism between calcium and bicarbonate

28 July 2018

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CO(2)/HCO(3)(-)-responsive soluble adenylyl cyclase as a putative metabolic sensor

28 July 2018

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Identification and functional analysis of splice variants of the germ cell soluble adenylyl cyclase

28 July 2018

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Regulation and role of adenylyl cyclase isoforms

28 July 2018

1 reference

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28 July 2018

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28 July 2018

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Two-metal-Ion catalysis in adenylyl cyclase

28 July 2018

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28 July 2018

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Cytosolic adenylyl cyclase defines a unique signaling molecule in mammals

28 July 2018

1 reference

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Crystal structure of the catalytic domains of adenylyl cyclase in a complex with Gsalpha.GTPgammaS

28 July 2018

1 reference

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Fluorescent guanine nucleotide analogs and G protein activation.

28 July 2018

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Mechanism of inhibition of HIV-1 reverse transcriptase by non-nucleoside inhibitors

28 July 2018

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Inhibition of the soluble form of testis adenylate cyclase by catechol estrogens and other catechols

28 July 2018

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28 July 2018

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Structural basis for the inhibition of mammalian membrane adenylyl cyclase by 2 '(3')-O-(N-Methylanthraniloyl)-guanosine 5 '-triphosphate

31 October 2018

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Direct inhibition of type 5 adenylyl cyclase prevents myocardial apoptosis without functional deterioration

31 October 2018

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31 October 2018

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Inhibition of adenylyl cyclase by acyclic nucleoside phosphonate antiviral agents

31 October 2018

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12 December 2020

Mechanism of nucleotide release from Rho by the GDP dissociation stimulator protein

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12 December 2020

Isoform-specific regulation of adenylyl cyclase by oxidized catecholamines

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12 December 2020

Kinetic Analysis of Interaction of Eukaryotic Release Factor 3 with Guanine Nucleotides

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12 December 2020

Identifiers

DOI

10.1021/JM800481Q

1 reference

26 July 2017

1 reference

26 July 2017

1 reference