Discovery of novel nuclear receptor modulating ligands: an integral role for peptide interaction profiling (Q33207350)

23 July 2017

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title

Discovery of novel nuclear receptor modulating ligands: an integral role for peptide interaction profiling (English)

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23 July 2017

Kenneth H Pearce

1

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23 July 2017

Marie A Iannone

series ordinal

2

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23 July 2017

Catherine A Simmons

series ordinal

3

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23 July 2017

John G Gray

series ordinal

4

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23 July 2017

1 September 2004

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23 July 2017

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23 July 2017

9

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23 July 2017

17

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23 July 2017

741-751

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A unified nomenclature system for the nuclear receptor superfamily

23 July 2017

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Steroid hormone receptors: evolution, ligands, and molecular basis of biologic function.

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https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Drug discovery: a historical perspective

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https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Genomics versus orphan nuclear receptors--a half-time report

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https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Activation functions 1 and 2 of nuclear receptors: molecular strategies for transcriptional activation

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Solution structure of the glucocorticoid receptor DNA-binding domain

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https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

The crystal structure of the estrogen receptor DNA-binding domain bound to DNA: how receptors discriminate between their response elements

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

The nuclear receptor ligand-binding domain: structure and function.

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Crystal structure of the ligand-binding domain of the human nuclear receptor RXR-alpha

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Ligand binding and co-activator assembly of the peroxisome proliferator-activated receptor-gamma

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Crystal structure of the glucocorticoid receptor ligand binding domain reveals a novel mode of receptor dimerization and coactivator recognition

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

A signature motif in transcriptional co-activators mediates binding to nuclear receptors

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Minireview: nuclear receptor coactivators--an update

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Molecular basis of agonism and antagonism in the oestrogen receptor

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

A structural biologist's view of the oestrogen receptor.

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Structure of the ligand-binding domain of oestrogen receptor beta in the presence of a partial agonist and a full antagonist

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Structural insights into the mode of action of a pure antiestrogen

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

The three-dimensional structures of antagonistic and agonistic forms of the glucocorticoid receptor ligand-binding domain: RU-486 induces a transconformation that leads to active antagonism

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Coregulator function: a key to understanding tissue specificity of selective receptor modulators

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Effects of tamoxifen on bone mineral density in postmenopausal women with breast cancer

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Tamoxifen activation of the estrogen receptor/AP-1 pathway: potential origin for the cell-specific estrogen-like effects of antiestrogens

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Coactivator and corepressor regulation of the agonist/antagonist activity of the mixed antiestrogen, 4-hydroxytamoxifen.

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Molecular determinants for the tissue specificity of SERMs

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Identification of a negative regulatory surface within estrogen receptor alpha provides evidence in support of a role for corepressors in regulating cellular responses to agonists and antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Differential SERM effects on corepressor binding dictate ERalpha activity in vivo

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Correlation between in vitro peptide binding profiles and cellular activities for estrogen receptor-modulating compounds.

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

The partial agonist activity of antagonist-occupied steroid receptors is controlled by a novel hinge domain-binding coactivator L7/SPA and the corepressors N-CoR or SMRT

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

RU486-induced glucocorticoid receptor agonism is controlled by the receptor N terminus and by corepressor binding

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Molecular control of immune/inflammatory responses: interactions between nuclear factor-kappa B and steroid receptor-signaling pathways

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Anti-inflammatory actions of glucocorticoids: molecular mechanisms

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Estrogen receptor-mediated cross-talk with growth factor signaling pathways

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

RETRACTED: Estrogen receptor-interacting protein that modulates its nongenomic activity-crosstalk with Src/Erk phosphorylation cascade

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Nongenomic actions of steroid hormones

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https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

3-[4-(1,2-Diphenylbut-1-enyl)phenyl]acrylic acid: a non-steroidal estrogen with functional selectivity for bone over uterus in rats

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

A novel antiinflammatory maintains glucocorticoid efficacy with reduced side effects

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Phage display for selection of novel binding peptides

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Selection of estrogen receptor beta- and thyroid hormone receptor beta-specific coactivator-mimetic peptides using recombinant peptide libraries

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https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Peptide antagonists of the human estrogen receptor

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https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Estrogen receptor (ER) modulators each induce distinct conformational changes in ER alpha and ER beta.

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Elucidation of the molecular mechanism of action of selective estrogen receptor modulators

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7 January 2021

T7 phage display: a novel genetic selection system for cloning RNA-binding proteins from cDNA libraries

1 reference

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7 January 2021

Probing protein conformational changes in living cells by using designer binding proteins: application to the estrogen receptor

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Kinetic, equilibrium, and thermodynamic analysis of macromolecular interactions with BIACORE.

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Hierarchical affinities and a bipartite interaction model for estrogen receptor isoforms and full-length steroid receptor coactivator (SRC/p160) family members

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Use of homogeneous time-resolved fluorescence energy transfer in the measurement of nuclear receptor activation

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Multiplexed molecular interactions of nuclear receptors using fluorescent microspheres

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Multiplexed microsphere-based flow cytometric assays

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Identification of selective estrogen receptor modulators by their gene expression fingerprints

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Identification, classification, and partial characterization of genes in humans and other vertebrates homologous to a fish membrane progestin receptor

1 reference

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7 January 2021

Rapid Signaling of Estrogen in Hypothalamic Neurons Involves a Novel G-Protein-Coupled Estrogen Receptor that Activates Protein Kinase C

1 reference

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7 January 2021

Receptor profiling and endocrine interactions of tibolone

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Selective estrogen receptor modulators

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Estrogen and selective estrogen receptor modulators: neuroprotection in the Women's Health Initiative era.

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

New Glucocorticosteroids with an improved therapeutic ratio?

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Eplerenone: cardiovascular protection

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Thiazolidinedione use, fluid retention, and congestive heart failure: a consensus statement from the American Heart Association and American Diabetes Association. October 7, 2003.

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Peroxisome proliferator-activated receptor-γ agonists in atherosclerosis: current evidence and future directions

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

The Use of Phage Display Technique for the Isolation of Androgen Receptor Interacting Peptides with (F/W)XXL(F/W) and FXXLY New Signature Motifs

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

Evaluation of ligand-dependent changes in AR structure using peptide probes

1 reference

https://api.crossref.org/works/10.1016%2FS1359-6446%2804%2903201-5

7 January 2021

10.1016/S1359-6446(04)03201-5

Identifiers

DOI

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23 July 2017

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