Constitutive activity at serotonin 5-HT(1D) receptors: detection by homologous GTPgammaS versus [(35)S]-GTPgammaS binding isotherms. (Q31561831)

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2 November 2019

title

Constitutive activity at serotonin 5-HT(1D) receptors: detection by homologous GTPgammaS versus [(35)S]-GTPgammaS binding isotherms (English)

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2 November 2019

author

Adrian Newman-Tancredi

series ordinal

2

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2 November 2019

author name string

V Audinot

series ordinal

1

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2 November 2019

M J Millan

series ordinal

3

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2 November 2019

publication date

1 January 2001

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2 November 2019

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2 November 2019

volume

40

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2 November 2019

issue

1

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2 November 2019

page(s)

57-64

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Binding profile of the novel 5-HT1B/1D receptor antagonist, [3H]GR 125,743, in guinea-pig brain: a comparison with [3H]5-carboxamidotryptamine

2 November 2019

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The selective 5-HT1B receptor inverse agonist 1'-methyl-5-[[2'-methyl-4'-(5-methyl-1,2, 4-oxadiazol-3-yl)biphenyl-4-yl]carbonyl]-2,3,6,7-tetrahydro- spiro[furo[2,3-f]indole-3,4'-piperidine] (SB-224289) potently blocks terminal 5-HT autoreceptor func

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Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a [35S]GTPgammaS binding study

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Labelling of recombinant human and native rat serotonin 5-HT1A receptors by a novel, selective radioligand, [3H]-S 15535: definition of its binding profile using agonists, antagonists and inverse agonists

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7 January 2021

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Pharmacological characterisation of [35S]-GTPgammaS binding to Chinese hamster ovary cell membranes stably expressing cloned human 5-HT1D receptor subtypes

7 January 2021

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10.1016/S0028-3908(00)00104-0

7 January 2021

Identifiers

DOI

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2 November 2019

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