Structural determinants of efficacy at A3 adenosine receptors: modification of the ribose moiety. (Q30431164)

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27 December 2019

title

Structural determinants of efficacy at A3 adenosine receptors: modification of the ribose moiety (English)

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13

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Juan B. Rodríguez

12

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1

Zhan-Guo Gao

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Ariel S Gross

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Lak Shin Jeong

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3

Hyung Ryong Moon

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Dae Hong Shin

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Neli Melman

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Liaman Mamedova

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author name string

Hea Ok Kim

4

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Won Jun Choi

5

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Eleonora Elhalem

7

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Maria J Comin

8

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language of work or name

English

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publication date

1 March 2004

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27 December 2019

published in

Biochemical Pharmacology

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volume

67

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page(s)

893-901

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issue

5

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Some quantitative uses of drug antagonists

27 December 2019

cites work

1 reference

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Behavioral characterization of mice lacking the A3 adenosine receptor: sensitivity to hypoxic neurodegeneration

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28 July 2018

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A3adenosine receptor agonist IB-MECA reduces myocardial ischemia-reperfusion injury in dogs

28 July 2018

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Stereoselective synthesis of a novel apio analogue of neplanocin A as potential S-adenosylhomocysteine hydrolase inhibitor

28 July 2018

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Identification by site-directed mutagenesis of residues involved in ligand recognition and activation of the human A3 adenosine receptor

28 July 2018

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28 July 2018

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5'-O-alkyl ethers of N,2-substituted adenosine derivatives: partial agonists for the adenosine A1 and A3 receptors

28 July 2018

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A(1) or A(3) adenosine receptors induce late preconditioning against infarction in conscious rabbits by different mechanisms

28 July 2018

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Distinct cardioprotective effects of adenosine mediated by differential coupling of receptor subtypes to phospholipases C and D.

28 July 2018

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N6,5'-Disubstituted adenosine derivatives as partial agonists for the human adenosine A3 receptor

28 July 2018

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125I-4-aminobenzyl-5'-N-methylcarboxamidoadenosine, a high affinity radioligand for the rat A3 adenosine receptor

28 July 2018

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Structure-activity relationships of N6-benzyladenosine-5'-uronamides as A3-selective adenosine agonists

28 July 2018

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Adenosine A3 receptor stimulation and cerebral ischemia

28 July 2018

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

28 July 2018

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Molecular cloning and characterization of an adenosine receptor: the A3 adenosine receptor

28 July 2018

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A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

28 July 2018

1 reference

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Design, synthesis and binding affinity of 3'-fluoro analogues of Cl-IB-MECA as adenosine A3 receptor ligands

28 July 2018

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A3 adenosine receptor knockout mice are protected against ischemia- and myoglobinuria-induced renal failure

26 November 2018

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Structural determinants of A(3) adenosine receptor activation: nucleoside ligands at the agonist/antagonist boundary

26 November 2018

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Knockout of A3 adenosine receptors reduces mouse intraocular pressure

26 November 2018

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N(6)-alkyl-2-alkynyl derivatives of adenosine as potent and selective agonists at the human adenosine A(3) receptor and a starting point for searching A(2B) ligands

26 November 2018

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2-Chloro-N(6)-cyclopentyladenosine, adenosine A(1) receptor agonist, antagonizes the adenosine A(3) receptor

26 November 2018

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A physiological role of the adenosine A3 receptor: sustained cardioprotection

26 November 2018

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Protective effects of renal ischemic preconditioning and adenosine pretreatment: role of A(1) and A(3) receptors

26 November 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/15104242

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12 December 2020

based on heuristic

N6-[2-(3,5-dimethoxyphenyl)-2-(2-methylphenyl)ethyl]adenosine and its uronamide derivatives. Novel adenosine agonists with both high affinity and high selectivity for the adenosine A2 receptor

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/15104242

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

A modification of a protein-binding method for rapid quantification of cAMP in cell-culture supernatants and body fluid

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/15104242

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.BCP.2003.10.006

1 reference

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27 December 2019

1 reference

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27 December 2019

1 reference