Label-free integrative pharmacology on-target of opioid ligands at the opioid receptor family (Q28709650)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23497702%20AND%20SRC:MED&resulttype=core&format=json

26 February 2020

title

Label-free integrative pharmacology on-target of opioid ligands at the opioid receptor family (English)

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26 February 2020

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4

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26 February 2020

author name string

Megan Morse

1

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26 February 2020

Haiyan Sun

2

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26 February 2020

Elizabeth Tran

3

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26 February 2020

Ye Fang

5

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26 February 2020

language of work or name

English

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publication date

12 March 2013

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BMC pharmacology & toxicology

26 February 2020

published in

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26 February 2020

volume

14

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26 February 2020

issue

1

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page(s)

17

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Ligand-directed functional selectivity at the mu opioid receptor revealed by label-free integrative pharmacology on-target

26 February 2020

cites work

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17 March 2017

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17 March 2017

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Oligomerization of opioid receptors with beta 2-adrenergic receptors: a role in trafficking and mitogen-activated protein kinase activation

17 March 2017

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17 March 2017

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17 March 2017

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Comprehensive analysis of kinase inhibitor selectivity

17 March 2017

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The potential for selective pharmacological therapies through biased receptor signaling

7 April 2017

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Label-free integrative pharmacology on-target of drugs at the β(2)-adrenergic receptor

3 June 2018

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Dynamic mass redistribution assays decode surface influence on signaling of endogenous purinergic P2Y receptors.

3 June 2018

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Functional selectivity at the μ-opioid receptor: implications for understanding opioid analgesia and tolerance.

3 June 2018

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Opioid receptor subtypes: fact or artifact?

3 June 2018

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Label-Free Receptor Assays

3 June 2018

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PROBING CANCER SIGNALING WITH RESONANT WAVEGUIDE GRATING BIOSENSORS

3 June 2018

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Label-free whole-cell assays: expanding the scope of GPCR screening

3 June 2018

1 reference

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Being mindful of seven-transmembrane receptor 'guests' when assessing agonist selectivity

3 June 2018

1 reference

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Kinase cascades and ligand-directed signaling at the kappa opioid receptor

3 June 2018

1 reference

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Seven transmembrane receptors as shapeshifting proteins: the impact of allosteric modulation and functional selectivity on new drug discovery

3 June 2018

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Visualization of omics data for systems biology

3 June 2018

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Opioid-receptor-heteromer-specific trafficking and pharmacology

3 June 2018

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Cellular assays as portals to seven-transmembrane receptor-based drug discovery

3 June 2018

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Label-free optical biosensor for probing integrative role of adenylyl cyclase in G protein-coupled receptor signaling

3 June 2018

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Evaluating cellular impedance assays for detection of GPCR pleiotropic signaling and functional selectivity

3 June 2018

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On the fitting of binding data when receptor dimerization is suspected

3 June 2018

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Label-free optical biosensor for ligand-directed functional selectivity acting on beta(2) adrenoceptor in living cells.

3 June 2018

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The evasive nature of drug efficacy: implications for drug discovery

3 June 2018

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GPCR functional selectivity has therapeutic impact

3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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3 June 2018

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Diversity and complexity of the mu opioid receptor gene: alternative pre-mRNA splicing and promoters

3 June 2018

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New concepts in drug discovery: collateral efficacy and permissive antagonism

3 June 2018

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A role for heterodimerization of mu and delta opiate receptors in enhancing morphine analgesia

3 June 2018

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Regulation of opioid receptor trafficking and morphine tolerance by receptor oligomerization

3 June 2018

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A delta opioid receptor lacking the third cytoplasmic loop is generated by atypical mRNA processing in human malignomas

3 June 2018

1 reference

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Molecular mechanisms and regulation of opioid receptor signaling

3 June 2018

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Type-specific sorting of G protein-coupled receptors after endocytosis

3 June 2018

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International Union of Pharmacology. XII. Classification of opioid receptors.

3 June 2018

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Differential regulation of mu and delta opiate receptors by morphine, selective agonists and antagonists and differentiating agents in SH-SY5Y human neuroblastoma cells

3 June 2018

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ADP-ribosyltransferase mutations in the catalytic S-1 subunit of pertussis toxin

3 June 2018

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Comparative pharmacological properties and functional coupling of mu and delta opioid receptor sites in human neuroblastoma SH-SY5Y cells

3 June 2018

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Regulation of cyclic AMP by the mu-opioid receptor in human neuroblastoma SH-SY5Y cells.

3 June 2018

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ADP-ribosylation of membrane proteins catalyzed by cholera toxin: basis of the activation of adenylate cyclase

3 June 2018

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Differential regulation of the human kappa opioid receptor by agonists: etorphine and levorphanol reduced dynorphin A- and U50,488H-induced internalization and phosphorylation

3 June 2018

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Crossref

https://api.crossref.org/works/10.1186%2F2050-6511-14-17

The development of label-free cellular assays for drug discovery

21 January 2018

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Functional selectivity of G protein signaling by agonist peptides and thrombin for the protease-activated receptor-1.

21 January 2018

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21 January 2018

Identifiers

DOI

10.1186/2050-6511-14-17

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23497702%20AND%20SRC:MED&resulttype=core&format=json

Dimensions Publication ID

26 February 2020

0 references

1 reference

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26 February 2020

PubMed publication ID

23497702

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23497702%20AND%20SRC:MED&resulttype=core&format=json