Discovery of epigenetic regulator I-BET762: lead optimization to afford a clinical candidate inhibitor of the BET bromodomains (Q27685477)

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Discovery of epigenetic regulator I-BET762: lead optimization to afford a clinical candidate inhibitor of the BET bromodomains
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    Discovery of epigenetic regulator I-BET762: lead optimization to afford a clinical candidate inhibitor of the BET bromodomains (English)
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    Romain Gosmini
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    Jérôme Toum
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    Catherine A Clément
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    Mélanie Barnathan
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    Jean-Marie Brusq
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    Jacqueline E Mordaunt
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    Richard M Grimes
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    Miriam Crowe
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    Olivier Pineau
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    Myriam Ajakane
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    Alain Daugan
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    Phillip Jeffrey
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    Leanne Cutler
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    Andrea C Haynes
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    Nicholas N Smithers
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    Chun-wa Chung
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    Antonia Lewis
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    Jason Witherington
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    Nigel Parr
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    Rab K Prinjha
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    Edwige Nicodème
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    10 October 2013
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    56
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    7501-15
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    19
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