Lead optimization of a 4-aminopyridine benzamide scaffold to identify potent, selective, and orally bioavailable TYK2 inhibitors (Q27684603)

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Lead optimization of a 4-aminopyridine benzamide scaffold to identify potent, selective, and orally bioavailable TYK2 inhibitors
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    Lead optimization of a 4-aminopyridine benzamide scaffold to identify potent, selective, and orally bioavailable TYK2 inhibitors (English)
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    Jun Liang
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    Kathy Barrett
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    Leo Berezhkovsky
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    Wade Blair
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    Christine Chang
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    Donnie Delarosa
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    Jim Driscoll
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    Paul Gibbons
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    Jason Halladay
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    Adam Johnson
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    Pawan Bir Kohli
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    Yingjie Lai
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    Yanzhou Liu
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    Joseph Lyssikatos
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    Priscilla Mantik
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    Kapil Menghrajani
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    Jeremy Murray
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    Ivan Peng
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    Amy Sambrone
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    Steven Shia
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    Young Shin
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    Jan Smith
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    Sue Sohn
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    Vickie Tsui
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    Lawren C Wu
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    Yisong Xiao
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    Wenqian Yang
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    Judy Young
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    Birong Zhang
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    Bing-yan Zhu
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    Steven Magnuson
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    13 June 2013
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    56
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    11
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    4521-36
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