Discovery of 5-chloro-N2-[(1S)-1-(5-fluoropyrimidin-2-yl)ethyl]-N4-(5-methyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine (AZD1480) as a novel inhibitor of the Jak/Stat pathway (Q27666212)

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Discovery of 5-chloro-N2-[(1S)-1-(5-fluoropyrimidin-2-yl)ethyl]-N4-(5-methyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine (AZD1480) as a novel inhibitor of the Jak/Stat pathway
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    Discovery of 5-chloro-N2-[(1S)-1-(5-fluoropyrimidin-2-yl)ethyl]-N4-(5-methyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine (AZD1480) as a novel inhibitor of the Jak/Stat pathway (English)
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    Stephanos Ioannidis
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    Michelle L Lamb
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    Tao Wang
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    Lynsie Almeida
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    Michael H Block
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    Audrey M Davies
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    Bo Peng
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    Mei Su
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    Hai-Jun Zhang
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    Ethan Hoffmann
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    Caroline Rivard
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    Isabelle Green
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    Tina Howard
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    Hannah Pollard
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    Jon Read
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    Marat Alimzhanov
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    Geraldine Bebernitz
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    Kirsten Bell
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    Minwei Ye
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    Dennis Huszar
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    Michael Zinda
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    13 January 2011
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    54
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    1
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    262-76
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