Conserved Binding Mode of Human β 2 Adrenergic Receptor Inverse Agonists and Antagonist Revealed by X-ray Crystallography (Q27663654)

4

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Daniel Wacker

1

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Vadim Cherezov

6

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Ruben Abagyan

5

object named as

Ruben Abagyan

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Raymond C. Stevens

object named as

Raymond C Stevens

7

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Gustavo Fenalti

2

object named as

Gustavo Fenalti

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author name string

Monica A Brown

Journal of the American Chemical Society

3

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language of work or name

English

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publication date

25 August 2010

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published in

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volume

132

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page(s)

11443-5

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issue

33

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cites work

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Structure of a beta1-adrenergic G-protein-coupled receptor

20 March 2017

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A Specific Cholesterol Binding Site Is Established by the 2.8 Å Structure of the Human β2-Adrenergic Receptor

20 March 2017

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High-resolution crystal structure of an engineered human beta2-adrenergic G protein-coupled receptor

20 March 2017

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Dynamics of the beta2-adrenergic G-protein coupled receptor revealed by hydrogen-deuterium exchange

20 March 2017

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Ligand and structure-based models for the prediction of ligand-receptor affinities and virtual screenings: Development and application to the beta(2)-adrenergic receptor

29 September 2017

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The effect of ligand efficacy on the formation and stability of a GPCR-G protein complex

29 September 2017

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Analysis of full and partial agonists binding to beta2-adrenergic receptor suggests a role of transmembrane helix V in agonist-specific conformational changes

29 September 2017

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Structure-based discovery of beta2-adrenergic receptor ligands

29 September 2017

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Identifying conformational changes of the beta(2) adrenoceptor that enable accurate prediction of ligand/receptor interactions and screening for GPCR modulators

29 September 2017

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High-resolution distance mapping in rhodopsin reveals the pattern of helix movement due to activation

29 September 2017

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Analysis of hydrophobic interactions of antagonists with the beta2-adrenergic receptor

29 September 2017

1 reference

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Insights into signaling from the β2-adrenergic receptor structure

27 November 2018

1 reference

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Plasmon-waveguide resonance studies of ligand binding to the human beta 2-adrenergic receptor

27 November 2018

1 reference

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27 November 2018

Identifiers

DOI

10.1021/JA105108Q

1 reference

499161

499161

1 reference

1 reference

1 reference